| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5248912 | B | Inhibition of NTMT1 (unknown origin) using SPKRIAKRRS(CONH2) peptide as substrate assessed as SAH production incubated for 10 mins in the presence of SAM by HPLC analysis | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 2. | ALA5248913 | B | Potency index, ratio of DC541 IC50 to test compound IC50 for inhibition of NTMT1 (unknown origin) using SPKRIAKRRS(CONH2) peptide as substrate assessed as SAH production incubated for 10 mins in the presence of SAM by HPLC analysis | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 3. | ALA5248914 | B | PROTAC activity at VHL/NTMT1 in human HCT-116 cells assessed as reduction in NTMT1 protein level incubated for 24 hrs by Western blot analysis | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 4. | ALA5248915 | B | PROTAC activity at VHL/NTMT1 in human HT-29 cells assessed as reduction in NTMT1 protein level incubated for 24 hrs by Western blot analysis | Homo sapiens | 3 | cell-based format | Scientific Literature |
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