| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5264691 | A | Metabolic stability in dog liver microsomes assessed as intrinsic clearance | Canis lupus familiaris | 1 | ALA5260843 | microsome format | Scientific Literature | |
| 2. | ALA5264692 | A | Metabolic stability in rat liver microsomes assessed as intrinsic clearance | Rattus norvegicus | 1 | ALA5260843 | microsome format | Scientific Literature | |
| 3. | ALA5264693 | A | Metabolic stability in human liver microsomes assessed as intrinsic clearance | Homo sapiens | 1 | ALA5260843 | microsome format | Scientific Literature | |
| 4. | ALA5264703 | F | Induction of ROS generation in human MGC-803 cells at 3 uM incubated for 24 hrs by DCFH-DA staining based flow cytometry analysis (Rvb = 2.2%) | Homo sapiens | 1 | ALA5260843 | cell-based format | Scientific Literature | |
| 5. | ALA5264704 | F | Induction of ROS generation in human MGC-803 cells at 1 uM incubated for 24 hrs by DCFH-DA staining based flow cytometry analysis (Rvb = 2.2%) | Homo sapiens | 1 | ALA5260843 | cell-based format | Scientific Literature | |
| 6. | ALA5264705 | F | Induction of ROS generation in human MGC-803 cells at 0.3 uM incubated for 24 hrs by DCFH-DA staining based flow cytometry analysis (Rvb = 2.2%) | Homo sapiens | 1 | ALA5260843 | cell-based format | Scientific Literature | |
| 7. | ALA5264707 | B | Inhibition of cullin5 neddylation in human KYSE-70 cells at 0.3 to 10 uM incubated for 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA5260843 | cell-based format | Scientific Literature | |
| 8. | ALA5264708 | B | Inhibition of cullin4B neddylation in human KYSE-70 cells at 0.3 to 10 uM incubated for 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA5260843 | cell-based format | Scientific Literature | |
| 9. | ALA5264709 | B | Inhibition of cullin4A neddylation in human KYSE-70 cells at 0.3 to 10 uM incubated for 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA5260843 | cell-based format | Scientific Literature | |
| 10. | ALA5264710 | B | Inhibition of cullin2 neddylation in human KYSE-70 cells at 0.3 to 10 uM incubated for 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA5260843 | cell-based format | Scientific Literature | |
| 11. | ALA5264711 | B | Inhibition of cullin3 neddylation in human KYSE-70 cells incubated for 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA5260843 | cell-based format | Scientific Literature | |
| 12. | ALA5264714 | B | Inhibition of cullin5 neddylation in UBC/DCN1 overactivated human MGC-803 cells at 0.3 to 10 uM incubated for 24 hrs by Western blot analysis | Homo sapiens | 3 | ALA5260843 | cell-based format | Scientific Literature | |
| 13. | ALA5264715 | B | Inhibition of cullin4B neddylation in UBC/DCN1 overactivated human MGC-803 cells at 0.3 to 10 uM incubated for 24 hrs by Western blot analysis | Homo sapiens | 3 | ALA5260843 | cell-based format | Scientific Literature | |
| 14. | ALA5264716 | B | Inhibition of cullin4A neddylation in UBC/DCN1 overactivated human MGC-803 cells at 0.3 to 10 uM incubated for 24 hrs by Western blot analysis | Homo sapiens | 3 | ALA5260843 | cell-based format | Scientific Literature | |
| 15. | ALA5264717 | B | Inhibition of cullin2 neddylation in UBC/DCN1 overactivated human MGC-803 cells at 0.3 to 10 uM incubated for 24 hrs by Western blot analysis | Homo sapiens | 3 | ALA5260843 | cell-based format | Scientific Literature | |
| 16. | ALA5264718 | B | Inhibition of cullin1 neddylation in UBC/DCN1 overactivated human MGC-803 cells at 10 uM incubated for 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA5260843 | cell-based format | Scientific Literature | |
| 17. | ALA5264719 | B | Inhibition of cullin3 neddylation in UBC/DCN1 overactivated human MGC-803 cells at 3 uM incubated for 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA5260843 | cell-based format | Scientific Literature | |
| 18. | ALA5264727 | B | Binding affinity to DCN1 in human MGC-803 cells assessed as thermal stabilization incubated for 1 hr followed by heating at 53 degreeC for 3 mins by CETSA assay | Homo sapiens | 2 | ALA5260843 | cell-based format | Scientific Literature | |
| 19. | ALA5264728 | B | Reversible inhibition of GST-tagged DCN1 PONY domain (unknown origin)/human N-terminal acetylated UBC12 (1 to 12 residues) protein-protein interaction at 500 nM preincubated for 1 hr followed by Ac-UBC12-biotin addition by HTRF based ultrafiltration analysis | Homo sapiens | 2 | ALA5260843 | protein format | Scientific Literature | |
| 20. | ALA5264729 | B | Reversible inhibition of GST-tagged DCN1 PONY domain (unknown origin)/human N-terminal acetylated UBC12 (1 to 12 residues) protein-protein interaction at 500 nM preincubated for 1 hr followed by Ac-UBC12-biotin addition by HTRF based dilution analysis | Homo sapiens | 2 | ALA5260843 | protein format | Scientific Literature |
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