# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA5261606 | Binding | Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | ALA5260810 | single protein format | Scientific Literature | |
2. | ALA5261607 | Binding | Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | ALA5260810 | single protein format | Scientific Literature | |
3. | ALA5261609 | Binding | Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | ALA5260810 | single protein format | Scientific Literature | |
4. | ALA5261611 | Binding | Displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | ALA5260810 | single protein format | Scientific Literature | |
5. | ALA5261613 | Binding | Displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | ALA5260810 | single protein format | Scientific Literature | |
6. | ALA5261614 | Binding | Binding affinity to ZsGreen fused-BRD9 (M1 to T597 residues) (unknown origin) expressed in human U2OS-C433 cells assessed as induction of protein bromodomain localization from chromatin by measuring formation of large nuclear puncta by fluorescence based assay | Homo sapiens | 10 | ALA5260810 | cell-based format | Scientific Literature | |
7. | ALA5261635 | Binding | Inhibition of BRD9 in human PC-9 cells assessed as reduction in ALDH1A1 gene expression at 2 uM preincubated with erlotinib for 8 days followed by compound addition and measured after 24 hrs by RNA sequencing analysis | Homo sapiens | 1 | ALA5260810 | cell-based format | Scientific Literature | |
8. | ALA5261647 | Functional | Cytotoxicity against human NALM-6 cells measured after 8 days | Homo sapiens | 2 | ALA5260810 | cell-based format | Scientific Literature | |
9. | ALA5261648 | Functional | Cytotoxicity against human NCI-H2373 cells measured after 8 days | Homo sapiens | 3 | ALA5260810 | cell-based format | Scientific Literature | |
10. | ALA5261649 | Functional | Cytotoxicity against human NCI-H2405 cells measured after 8 days | Homo sapiens | 3 | ALA5260810 | cell-based format | Scientific Literature | |
11. | ALA5261650 | Functional | Cytotoxicity against human MV4-11 cells measured after 8 days | Homo sapiens | 3 | ALA5260810 | cell-based format | Scientific Literature | |
12. | ALA5261651 | Functional | Cytotoxicity against human NCI-H2228 cells measured after 8 days | Homo sapiens | 3 | ALA5260810 | cell-based format | Scientific Literature | |
13. | ALA5261652 | Functional | Cytotoxicity against human NCI-H226 cells measured after 8 days | Homo sapiens | 3 | ALA5260810 | cell-based format | Scientific Literature | |
14. | ALA5261653 | Functional | Cytotoxicity against human NOMO-1 cells measured after 8 days | Homo sapiens | 2 | ALA5260810 | cell-based format | Scientific Literature | |
15. | ALA5261654 | Functional | Cytotoxicity against human HCC1576 cells measured after 8 days | Homo sapiens | 2 | ALA5260810 | cell-based format | Scientific Literature | |
16. | ALA5261655 | Functional | Cytotoxicity against human AMO1 cells measured after 8 days | Homo sapiens | 3 | ALA5260810 | cell-based format | Scientific Literature | |
17. | ALA5261656 | Functional | Cytotoxicity against mouse BaF3 cells measured after 8 days | Mus musculus | 2 | ALA5260810 | cell-based format | Scientific Literature | |
18. | ALA5261657 | Functional | Cytotoxicity against human CA46 cells measured after 8 days | Homo sapiens | 3 | ALA5260810 | cell-based format | Scientific Literature | |
19. | ALA5261658 | Functional | Cytotoxicity against human Daudi cells measured after 8 days | Homo sapiens | 3 | ALA5260810 | cell-based format | Scientific Literature | |
20. | ALA5261659 | Functional | Cytotoxicity against human EB-3 cells measured after 8 days | Homo sapiens | 3 | ALA5260810 | cell-based format | Scientific Literature |