| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5238165 | B | Inhibition of FXIIa (unknown origin) using Ac-QRFR-pNA as substrate measured at 30 sec interval by microplate reader assay | Homo sapiens | 18 | ALA5236588 | assay format | Scientific Literature | |
| 2. | ALA5238166 | B | Potency index, ratio of M8 Ki to test compound Ki for inhibition of FXIIa (unknown origin) | Homo sapiens | 17 | ALA5236588 | assay format | Scientific Literature | |
| 3. | ALA5238168 | B | Inhibition of human cationic trypsin using Boc-VPR-MCA as susbtrate | Homo sapiens | 3 | ALA5236588 | assay format | Scientific Literature | |
| 4. | ALA5238169 | B | Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate | Homo sapiens | 3 | ALA5236588 | single protein format | Scientific Literature | |
| 5. | ALA5238170 | B | Inhibition of human FXa using Z-Pyr-GR-MCA as substrate | Homo sapiens | 3 | ALA5236588 | assay format | Scientific Literature | |
| 6. | ALA5238171 | B | Inhibition of human FXIa using Boc-Glu(OBzl)-AR-MCA as substrate | Homo sapiens | 3 | ALA5236588 | assay format | Scientific Literature | |
| 7. | ALA5238172 | B | Inhibition of human beta-FIXa using Boc-QGR-MCA as substrate | Homo sapiens | 3 | ALA5236588 | assay format | Scientific Literature | |
| 8. | ALA5238173 | B | Inhibition of human thrombin using Boc-VPR-MCA as substrate | Homo sapiens | 3 | ALA5236588 | single protein format | Scientific Literature | |
| 9. | ALA5238174 | B | Inhibition of human plasma kallikrein using Z-FR-MCA as substrate | Homo sapiens | 3 | ALA5236588 | cell-free format | Scientific Literature | |
| 10. | ALA5238175 | B | Inhibition of recombinant human matriptase using Boc-QAR-MCA as substrate | Homo sapiens | 3 | ALA5236588 | single protein format | Scientific Literature | |
| 11. | ALA5238176 | B | Inhibition of human cationic trypsin at 5 uM using Boc-VPR-MCA as susbtrate relative to control | Homo sapiens | 1 | ALA5236588 | assay format | Scientific Literature | |
| 12. | ALA5238177 | B | Inhibition of human plasmin at 5 uM using Ac-RM(O2)YR-pNA as substrate relative to control | Homo sapiens | 1 | ALA5236588 | single protein format | Scientific Literature | |
| 13. | ALA5238178 | B | Inhibition of human FXa at 5 uM using Z-Pyr-GR-MCA as substrate relative to control | Homo sapiens | 3 | ALA5236588 | assay format | Scientific Literature | |
| 14. | ALA5238179 | B | Inhibition of human FXIa at 5 uM using Boc-Glu(OBzl)-AR-MCA as substrate relative to control | Homo sapiens | 2 | ALA5236588 | assay format | Scientific Literature | |
| 15. | ALA5238180 | B | Inhibition of human beta-FIXa at 5 uM using Boc-QGR-MCA as substrate relative to control | Homo sapiens | 2 | ALA5236588 | assay format | Scientific Literature | |
| 16. | ALA5238181 | B | Inhibition of human thrombin at 5 uM using Boc-VPR-MCA as substrate relative to control | Homo sapiens | 2 | ALA5236588 | single protein format | Scientific Literature | |
| 17. | ALA5238182 | B | Inhibition of human plasma kallikrein at 5 uM using Z-FR-MCA as substrate relative to control | Homo sapiens | 2 | ALA5236588 | cell-free format | Scientific Literature | |
| 18. | ALA5238184 | A | Stability of compound in human serum at 50 uM incubated for 24 hrs by reversed phase HPLC analysis | Homo sapiens | 3 | ALA5236588 | cell-free format | Scientific Literature | |
| 19. | ALA5238185 | A | Stability of compound in human serum at 50 uM incubated for 8 hrs by reversed phase HPLC analysis | Homo sapiens | 1 | ALA5236588 | cell-free format | Scientific Literature | |
| 20. | ALA5238186 | F | Anticoagulant activity in human plasma assessed as prolongation of activated partial thromboplastin time by measuring concentration required to double aPTT | Homo sapiens | 1 | ALA5236588 | organism-based format | Scientific Literature |
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