| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5224961 | B | Antagonist activity at human P2Y6R expressed in human 1321N1 cells assessed as inhibition of UDP-induced calcium mobilization by FLIPR assay | Homo sapiens | 21 | ALA5223123 | cell-based format | Scientific Literature | |
| 2. | ALA5224965 | B | Antagonist activity at Meleagris P2Y1R expressed in human 1321N1 cells assessed as inhibition of UDP-induced calcium mobilization at 100 uM by FLIPR assay relative to control | Meleagris gallopavo | 5 | ALA5223123 | cell-based format | Scientific Literature | |
| 3. | ALA5224966 | B | Antagonist activity at human P2Y2R expressed in human 1321N1 cells assessed as inhibition of UDP-induced calcium mobilization at 100 uM by FLIPR assay relative to control | Homo sapiens | 5 | ALA5223123 | cell-based format | Scientific Literature | |
| 4. | ALA5224967 | B | Antagonist activity at human P2Y4R expressed in human 1321N1 cells assessed as inhibition of UDP-induced calcium mobilization at 100 uM by FLIPR assay relative to control | Homo sapiens | 5 | ALA5223123 | cell-based format | Scientific Literature | |
| 5. | ALA5224968 | B | Antagonist activity at mouse P2Y6R expressed in human 1321N1 cells assessed as inhibition of UDP-induced calcium mobilization by FLIPR assay | Mus musculus | 11 | ALA5223123 | cell-based format | Scientific Literature | |
| 6. | ALA5224970 | B | Selectivity ratio of IC50 for mouse P2Y6R to IC50 for human P2Y6R | 13 | ALA5223123 | assay format | Scientific Literature | ||
| 7. | ALA5224974 | B | Binding affinity to adrenergic alpha 2b receptor (unknown origin) | Homo sapiens | 1 | ALA5223123 | single protein format | Scientific Literature | |
| 8. | ALA5224975 | B | Binding affinity to adrenergic alpha 2c receptor (unknown origin) | Homo sapiens | 1 | ALA5223123 | single protein format | Scientific Literature | |
| 9. | ALA5224976 | B | Binding affinity to sigma 1 receptor (unknown origin) | Homo sapiens | 1 | ALA5223123 | single protein format | Scientific Literature | |
| 10. | ALA5224977 | B | Binding affinity to histamine H1 receptor (unknown origin) | Homo sapiens | 1 | ALA5223123 | single protein format | Scientific Literature | |
| 11. | ALA5224978 | B | Binding affinity to adrenergic beta 3 (unknown origin) | Homo sapiens | 1 | ALA5223123 | single protein format | Scientific Literature | |
| 12. | ALA5224979 | B | Binding affinity to 5-HT2A (unknown origin) | Homo sapiens | 1 | ALA5223123 | single protein format | Scientific Literature | |
| 13. | ALA5224980 | T | Cytotoxicity against HEK293 cells assessed as reduction in cell viability at 100 uM measured after 24 hrs by MTT assay relative to control | Homo sapiens | 5 | ALA5223123 | cell-based format | Scientific Literature |
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