| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5225629 | B | Inhibition of KIT (unknown origin) in presence of ATP | Homo sapiens | 4 | ALA5223162 | single protein format | Scientific Literature | |
| 2. | ALA5225630 | B | Inhibition of FLT3 (unknown origin) in presence of ATP | Homo sapiens | 4 | ALA5223162 | single protein format | Scientific Literature | |
| 3. | ALA5225631 | B | Inhibition of TrkA (unknown origin) in presence of ATP | Homo sapiens | 4 | ALA5223162 | single protein format | Scientific Literature | |
| 4. | ALA5225632 | A | Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate by LC-MS analysis | Homo sapiens | 3 | ALA5223162 | microsome format | Scientific Literature | |
| 5. | ALA5225633 | A | Permeability across apical to basolateral side in human Caco2 cells at 50 uM and measured after 120 mins by LC-MS analysis | Homo sapiens | 8 | ALA5223162 | cell-based format | Scientific Literature | |
| 6. | ALA5225634 | B | Binding affinity to recombinant human HPK1 (1 to 346 residues) expressed sf9 cells incubated for 1 hr by LanthaScreen assay | Homo sapiens | 18 | ALA5223162 | cell-based format | Scientific Literature | |
| 7. | ALA5225635 | B | Inhibition of human HPK1 in human Jurkat cells assessed as reduction in SLP76 phosphorylation incubated for 1 hr by HTRF assay | Homo sapiens | 14 | ALA5223162 | cell-based format | Scientific Literature | |
| 8. | ALA5225636 | A | Intrinsic clearance in human liver microsomes at 1 uM and measured upto 30 mins in presence of NADPH by LC-MS analysis | Homo sapiens | 13 | ALA5223162 | microsome format | Scientific Literature | |
| 9. | ALA5225644 | A | Inhibition of CYP3A4 in human liver microsomes using testosterone as substrate by LC-MS analysis | Homo sapiens | 4 | ALA5223162 | microsome format | Scientific Literature |
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