#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA5239751	B	Inhibition of BODIPY FL vindoline binding to recombinant human GST-tagged PXR LBD (111 to 434 residues) expressed in baculovirus infected insect cells incubated for 1 mins under shaking condition followed by 60 mins under dark condition by TR-FRET assay	Homo sapiens	92		cell-based format	Scientific Literature
2.	ALA5239752	B	Inhibition of BODIPY FL vindoline binding to recombinant human GST-tagged PXR LBD (111 to 434 residues) expressed in baculovirus infected insect cells at 10 uM incubated for 1 mins under shaking condition followed by 60 mins under dark condition by TR-FRET assay relative to control	Homo sapiens	78		cell-based format	Scientific Literature
3.	ALA5239757	B	Antagonist activity at human PXR in human HepG2 cells co-expressing luciferase gene under control of CYP3A4 promoter assessed as inhibition in rifampicin-induced receptor activation incubated for 24 hrs by luminescence based analysis	Homo sapiens	60		cell-based format	Scientific Literature
4.	ALA5239758	B	Antagonist activity at human PXR in human HepG2 cells co-expressing luciferase gene under control of CYP3A4 promoter assessed as inhibition in rifampicin-induced receptor activation at 10 uM incubated for 24 hrs by luminescence based analysis relative to control	Homo sapiens	60		cell-based format	Scientific Literature
5.	ALA5239759	B	Agonist activity at human PXR in human HepG2 cells co-expressing luciferase gene under control of CYP3A4 promoter assessed as transcriptional activation at 30 uM incubated for 24 hrs by luminescence based analysis	Homo sapiens	64		cell-based format	Scientific Literature
6.	ALA5239760	B	Inverse agonist activity at human PXR in human HepG2 cells co-expressing luciferase gene under control of CYP3A4 promoter assessed as inhibition in receptor basal activity at 30 uM incubated for 24 hrs by luminescence based analysis	Homo sapiens	49		cell-based format	Scientific Literature
7.	ALA5239762	B	Effect on mouse PXR activity by luciferase reporter assay	Mus musculus	2		single protein format	Scientific Literature
8.	ALA5239763	B	Effect on CAR activity in human HepG2 cells co-expressing luciferase gene under control of CYP3A4 promoter by luciferase reporter assay	Homo sapiens	2		cell-based format	Scientific Literature
9.	ALA5239764	B	Effect on FXR activity in GeneBLAzer FXR-UAS-bla HEK 293T cells by fluorescence based analysis	Homo sapiens	2		cell-based format	Scientific Literature
10.	ALA5239765	B	Effect on LXRalpha activity in GeneBLAzer LXRalpha-UAS-bla HEK 293T cells by fluorescence based analysis	Homo sapiens	2		cell-based format	Scientific Literature
11.	ALA5239766	B	Effect on VDR activity in GeneBLAzer VDR-UAS-bla HEK 293T cells by fluorescence based analysis	Homo sapiens	2		cell-based format	Scientific Literature
12.	ALA5239767	T	Cytotoxicity against HEK293T cells assessed as reduction in cell viability measured after 24 to 72 hrs by celltiter-glo luminescent cell viability assay	Homo sapiens	2		cell-based format	Scientific Literature
13.	ALA5239768	T	Cytotoxicity against human HepG2 cells assessed as reduction in cell viability measured after 24 to 72 hrs by celltiter-glo luminescent cell viability assay	Homo sapiens	2		cell-based format	Scientific Literature
14.	ALA5239769	T	Cytotoxicity against human Hepa1-6 cells assessed as reduction in cell viability measured after 24 to 72 hrs by celltiter-glo luminescent cell viability assay	Homo sapiens	2		cell-based format	Scientific Literature
15.	ALA5239770	T	Cytotoxicity against human HepaRG cells assessed as reduction in cell viability measured after 24 to 72 hrs by celltiter-glo luminescent cell viability assay	Homo sapiens	2		cell-based format	Scientific Literature