| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5225666 | B | Agonist activity at human SST2 receptor expressed in CHO-K1 cells assessed as inhibition of NKH477-induced intracellular cAMP accumulation incubated for 20 mins by HTRF assay | Homo sapiens | 30 | cell-based format | Scientific Literature | ||
| 2. | ALA5225667 | B | Agonist activity at human SST1 receptor expressed in CHO-K1 cells assessed as inhibition of NKH477-induced intracellular cAMP accumulation incubated for 20 mins by HTRF assay | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 3. | ALA5225668 | B | Agonist activity at human SST3 receptor expressed in CHO-K1 cells assessed as inhibition of NKH477-induced intracellular cAMP accumulation incubated for 20 mins by HTRF assay | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 4. | ALA5225669 | B | Agonist activity at human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of NKH477-induced intracellular cAMP accumulation incubated for 20 mins by HTRF assay | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 5. | ALA5225670 | B | Agonist activity at human SST5 receptor expressed in CHO-K1 cells assessed as inhibition of NKH477-induced intracellular cAMP accumulation incubated for 20 mins by HTRF assay | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 6. | ALA5225671 | B | Selectivity index, ratio of pEC50 for agonist activity at human SST1 receptor expressed in CHO-K1 cells to pEC50 for agonist activity at human SST2 receptor expressed in CHO-K1 cells | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 7. | ALA5225672 | B | Selectivity index, ratio of pEC50 for agonist activity at human SST3 receptor expressed in CHO-K1 cells to pEC50 for agonist activity at human SST2 receptor expressed in CHO-K1 cells | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 8. | ALA5225673 | B | Selectivity index, ratio of pEC50 for agonist activity at human SST4 receptor expressed in CHO-K1 cells to pEC50 for agonist activity at human SST2 receptor expressed in CHO-K1 cells | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 9. | ALA5225674 | B | Selectivity index, ratio of pEC50 for agonist activity at human SST5 receptor expressed in CHO-K1 cells to pEC50 for agonist activity at human SST2 receptor expressed in CHO-K1 cells | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 10. | ALA5225675 | T | Inhibition of hERG by fluorescence polarization assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 11. | ALA5225676 | A | Half life in human liver microsomes | Homo sapiens | 5 | microsome format | Scientific Literature | ||
| 12. | ALA5225677 | A | Half life in rat liver microsomes | Rattus norvegicus | 5 | microsome format | Scientific Literature |
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