| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5253113 | Binding | Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter analysis | Homo sapiens | 79 | ALA5252514 | cell-based format | Scientific Literature | |
| 2. | ALA5253114 | Binding | Selectivity ratio, ratio of Ki for human KOR to Ki for human NOP | Homo sapiens | 9 | ALA5252514 | assay format | Scientific Literature | |
| 3. | ALA5253115 | Binding | Selectivity ratio, ratio of Ki for human KOR to Ki for human DOR | Homo sapiens | 9 | ALA5252514 | assay format | Scientific Literature | |
| 4. | ALA5253116 | Binding | Selectivity ratio, ratio of Ki for human KOR to Ki for human MOR | Homo sapiens | 9 | ALA5252514 | assay format | Scientific Literature | |
| 5. | ALA5253118 | Binding | Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as ERK phosphorylation incubated for 2 hrs by Alphascreen surefire method | Homo sapiens | 9 | ALA5252514 | cell-based format | Scientific Literature | |
| 6. | ALA5253119 | Binding | Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production incubated for 30 mins by LANCE cAMP assay | Homo sapiens | 9 | ALA5252514 | cell-based format | Scientific Literature | |
| 7. | ALA5253120 | ADME | Metabolic stability in Wistar rat plasma assessed as half life by HPLC analysis | Rattus norvegicus | 28 | ALA5252514 | cell-free format | Scientific Literature |
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