| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5240449 | B | Inverse agonist activity at GST tagged human PPARgamma LBD (231 to 505 residues) expressed in Escherichia coli BL21(DE3) assessed as recruitment of fluorescein labeled corepressor NCOR2 Smrt-ID2 peptide to PPARgamma LBD incubated for 24 hrs by LanthaScreen TR-FRET assay | Homo sapiens | 25 | assay format | Scientific Literature | ||
| 2. | ALA5240450 | B | Inverse agonist activity at GST tagged human PPARgamma LBD (231 to 505 residues) expressed in Escherichia coli BL21(DE3) assessed as recruitment of fluorescein labeled corepressor NCOR2 Smrt-ID2 peptide to PPARgamma LBD by measuring maximum efficacy incubated for 24 hrs by LanthaScreen TR-FRET assay | Homo sapiens | 23 | assay format | Scientific Literature | ||
| 3. | ALA5240451 | B | Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation incubated for 6 to 18 hrs by Nano-Glo luciferase assay | Homo sapiens | 25 | cell-based format | Scientific Literature | ||
| 4. | ALA5240452 | B | Inverse agonist activity at human PPARgamma in human RT112/84 transfected with NLuc-fused FABP4 assessed as reduction in PPARgamma transactivation by measuring maximum efficacy incubated for 6 to 18 hrs by Nano-Glo luciferase assay | Homo sapiens | 19 | cell-based format | Scientific Literature |
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