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# Aladdin ID Assay Type Description Organism Compounds Reference BAO Format Source 1. ALA5251532 B Inhibition of G9a (unknown origin) Homo sapiens 7 ALA5247652 single protein format Scientific Literature 2. ALA5251533 B Inhibition of GLP (unknown origin) Homo sapiens 5 ALA5247652 single protein format Scientific Literature 3. ALA5251534 B Inhibition of N-terminal GST-tagged human recombinant G9a (785 to 1210 residues) expressed in baculovirus infected Sf9 cells incubated for 1 hr by AlphaLISA analysis Homo sapiens 57 ALA5247652 cell-based format Scientific Literature 4. ALA5251539 F Antiproliferative activity against human MOLT-4 cells assessed as inhibition of cell growth with replenishment of medium with compound on day 4 and 7 and measured after 12 days by ATPlite assay Homo sapiens 6 ALA5247652 cell-based format Scientific Literature 5. ALA5251541 F Downregulation of H3K9 dimethylation in human MOLT-4 cells at 1 uM by Western blot analysis Homo sapiens 2 ALA5247652 cell-based format Scientific Literature 6. ALA5251542 A Cmax in ICR mouse at 25 mg/kg, ip Mus musculus 2 ALA5247652 organism-based format Scientific Literature 7. ALA5251543 A AUC (0 to infinity) in ICR mouse at 25 mg/kg, ip Mus musculus 2 ALA5247652 organism-based format Scientific Literature 8. ALA5251544 A Tmax in ICR mouse at 25 mg/kg, ip Mus musculus 2 ALA5247652 organism-based format Scientific Literature 9. ALA5251545 A Half life in ICR mouse at 25 mg/kg, ip Mus musculus 2 ALA5247652 organism-based format Scientific Literature 10. ALA5251546 F Antitumor activity against DEN-induced human HCC tumor in C57BL/6 mouse at 20 to 50 mg/kg, ip measured after 48 weeks Homo sapiens 1 ALA5247652 organism-based format Scientific Literature 11. ALA5251547 T Toxicity in C57BL/6 mouse assessed as body weight loss at 20 to 50 mg/kg, ip measured after 48 weeks Mus musculus 1 ALA5247652 organism-based format Scientific Literature 12. ALA5251548 F Invivo inhibition of G9a in C57BL/6 mouse liver assessed as reduction in H3K9me2 level at 20 to 50 mg/kg, ip measured after 5 days by Westernblot analysis Mus musculus 1 ALA5247652 organism-based format Scientific Literature 13. ALA5251549 A Drug concentration in C57BL/6 mouse liver at 20 mg/kg, ip measured after 4 hrs Mus musculus 1 ALA5247652 organism-based format Scientific Literature 14. ALA5251550 A Drug concentration in C57BL/6 mouse liver at 50 mg/kg, ip measured after 4 hrs Mus musculus 1 ALA5247652 organism-based format Scientific Literature 15. ALA5251551 A Drug concentration in C57BL/6 mouse plasma at 20 mg/kg, ip measured after 4 hrs Mus musculus 1 ALA5247652 organism-based format Scientific Literature 16. ALA5251552 A Drug concentration in C57BL/6 mouse plasma at 50 mg/kg, ip measured after 4 hrs Mus musculus 1 ALA5247652 organism-based format Scientific Literature 17. ALA5251553 F Invivo inhibition of G9a in C57BL/6 mouse liver assessed as H3 histone methylation at 20 to 50 mg/kg, ip measured after 5 days by Westernblot analysis Mus musculus 1 ALA5247652 organism-based format Scientific Literature