#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA5239751	B	Inhibition of BODIPY FL vindoline binding to recombinant human GST-tagged PXR LBD (111 to 434 residues) expressed in baculovirus infected insect cells incubated for 1 mins under shaking condition followed by 60 mins under dark condition by TR-FRET assay	Homo sapiens	92		cell-based format	Scientific Literature
2.	ALA5239752	B	Inhibition of BODIPY FL vindoline binding to recombinant human GST-tagged PXR LBD (111 to 434 residues) expressed in baculovirus infected insect cells at 10 uM incubated for 1 mins under shaking condition followed by 60 mins under dark condition by TR-FRET assay relative to control	Homo sapiens	78		cell-based format	Scientific Literature
3.	ALA5239755	B	Inverse agonist activity at human PXR in human HepG2 cells co-expressing luciferase gene under control of CYP3A4 promoter assessed as inhibition of receptor basal activity incubated for 24 hrs by luminescence based analysis	Homo sapiens	40		cell-based format	Scientific Literature
4.	ALA5239756	B	Inverse agonist activity at human PXR in human HepG2 cells co-expressing luciferase gene under control of CYP3A4 promoter assessed as inhibition in receptor basal activity at 10 uM incubated for 24 hrs by luminescence based analysis relative to control	Homo sapiens	40		cell-based format	Scientific Literature
5.	ALA5239757	B	Antagonist activity at human PXR in human HepG2 cells co-expressing luciferase gene under control of CYP3A4 promoter assessed as inhibition in rifampicin-induced receptor activation incubated for 24 hrs by luminescence based analysis	Homo sapiens	60		cell-based format	Scientific Literature
6.	ALA5239758	B	Antagonist activity at human PXR in human HepG2 cells co-expressing luciferase gene under control of CYP3A4 promoter assessed as inhibition in rifampicin-induced receptor activation at 10 uM incubated for 24 hrs by luminescence based analysis relative to control	Homo sapiens	60		cell-based format	Scientific Literature
7.	ALA5239759	B	Agonist activity at human PXR in human HepG2 cells co-expressing luciferase gene under control of CYP3A4 promoter assessed as transcriptional activation at 30 uM incubated for 24 hrs by luminescence based analysis	Homo sapiens	64		cell-based format	Scientific Literature
8.	ALA5239762	B	Effect on mouse PXR activity by luciferase reporter assay	Mus musculus	2		single protein format	Scientific Literature
9.	ALA5239763	B	Effect on CAR activity in human HepG2 cells co-expressing luciferase gene under control of CYP3A4 promoter by luciferase reporter assay	Homo sapiens	2		cell-based format	Scientific Literature
10.	ALA5239764	B	Effect on FXR activity in GeneBLAzer FXR-UAS-bla HEK 293T cells by fluorescence based analysis	Homo sapiens	2		cell-based format	Scientific Literature
11.	ALA5239765	B	Effect on LXRalpha activity in GeneBLAzer LXRalpha-UAS-bla HEK 293T cells by fluorescence based analysis	Homo sapiens	2		cell-based format	Scientific Literature
12.	ALA5239766	B	Effect on VDR activity in GeneBLAzer VDR-UAS-bla HEK 293T cells by fluorescence based analysis	Homo sapiens	2		cell-based format	Scientific Literature
13.	ALA5239767	T	Cytotoxicity against HEK293T cells assessed as reduction in cell viability measured after 24 to 72 hrs by celltiter-glo luminescent cell viability assay	Homo sapiens	2		cell-based format	Scientific Literature
14.	ALA5239768	T	Cytotoxicity against human HepG2 cells assessed as reduction in cell viability measured after 24 to 72 hrs by celltiter-glo luminescent cell viability assay	Homo sapiens	2		cell-based format	Scientific Literature
15.	ALA5239769	T	Cytotoxicity against human Hepa1-6 cells assessed as reduction in cell viability measured after 24 to 72 hrs by celltiter-glo luminescent cell viability assay	Homo sapiens	2		cell-based format	Scientific Literature
16.	ALA5239770	T	Cytotoxicity against human HepaRG cells assessed as reduction in cell viability measured after 24 to 72 hrs by celltiter-glo luminescent cell viability assay	Homo sapiens	2		cell-based format	Scientific Literature