| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5261606 | B | Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 2. | ALA5261607 | B | Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 3. | ALA5261608 | B | Selectivity ratio of IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) to IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) | Homo sapiens | 4 | protein format | Scientific Literature | ||
| 4. | ALA5261609 | B | Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 5. | ALA5261610 | B | Selectivity ratio of IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 2 (unknown origin) to IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) | Homo sapiens | 3 | protein format | Scientific Literature | ||
| 6. | ALA5261611 | B | Displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 7. | ALA5261612 | B | Selectivity ratio of IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) to IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 8. | ALA5261613 | B | Displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 9. | ALA5261614 | B | Binding affinity to ZsGreen fused-BRD9 (M1 to T597 residues) (unknown origin) expressed in human U2OS-C433 cells assessed as induction of protein bromodomain localization from chromatin by measuring formation of large nuclear puncta by fluorescence based assay | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 10. | ALA5261615 | B | Selectivity ratio of IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) to IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) | Homo sapiens | 4 | assay format | Scientific Literature |
The page will load shortly, Thanks for your patience!