# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA5238047 | Binding | Protac activity at BRD4/VHL E3 ligase in human MDA-MB-231 cells assessed as decrease in BRD4 expression at 1 uM incubated for 8 hrs by Western blot analysis | Homo sapiens | 8 | ALA5236581 | cell-based format | Scientific Literature | |
2. | ALA5238048 | Binding | Protac activity at BRD4/VHL E3 ligase in human MDA-MB-231 cells assessed as decrease in BRD4 expression at 1 uM incubated for 16 hrs by Western blot analysis | Homo sapiens | 9 | ALA5236581 | cell-based format | Scientific Literature | |
3. | ALA5238049 | Binding | Protac activity at BRD4/VHL E3 ligase in human MDA-MB-231 cells assessed as decrease in BRD4 expression at 1 uM incubated for 24 hrs by Western blot analysis | Homo sapiens | 9 | ALA5236581 | cell-based format | Scientific Literature | |
4. | ALA5238050 | Binding | Protac activity at BRD4/VHL E3 ligase in human MDA-MB-231 cells assessed as decrease in BRD4 expression at 0.1 nM to 10 uM incubated for 8 hrs by Western blot analysis | Homo sapiens | 6 | ALA5236581 | cell-based format | Scientific Literature | |
5. | ALA5238051 | Binding | Protac activity at BRD4/VHL E3 ligase in human MDA-MB-231 cells assessed as decrease in BRD4 expression incubated for 8 hrs by Western blot analysis | Homo sapiens | 7 | ALA5236581 | cell-based format | Scientific Literature |