| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5238222 | B | Inhibition of CDK7 (unknown origin) assessed as phosphorylation of ULight 4EBP1 peptide substrate measured after 2 hrs by FRET-based LANCE Ultra KinSelect assay | Homo sapiens | 30 | ALA5236590 | single protein format | Scientific Literature | |
| 2. | ALA5238224 | B | Inhibition of CDK2 (unknown origin) assessed as phosphorylation of ULight 4EBP1 peptide substrate measured after 2 hrs by FRET-based LANCE Ultra KinSelect assay | Homo sapiens | 19 | ALA5236590 | single protein format | Scientific Literature | |
| 3. | ALA5238226 | B | Selectivity ratio of IC50 for CDK7 (unknown origin) to IC50 for CDK2 (unknown origin) | Homo sapiens | 17 | ALA5236590 | assay format | Scientific Literature | |
| 4. | ALA5238227 | B | Irreversible inhibition of CDK7 (unknown origin) assessed as activity measured after 3 hrs by jump dilution method | Homo sapiens | 1 | ALA5236590 | single protein format | Scientific Literature | |
| 5. | ALA5238228 | B | Inhibition of CDK1 (unknown origin) | Homo sapiens | 1 | ALA5236590 | single protein format | Scientific Literature | |
| 6. | ALA5238229 | B | Inhibition of CDK3 (unknown origin) | Homo sapiens | 1 | ALA5236590 | single protein format | Scientific Literature | |
| 7. | ALA5238230 | B | Inhibition of CDK5 (unknown origin) | Homo sapiens | 1 | ALA5236590 | single protein format | Scientific Literature | |
| 8. | ALA5238231 | B | Inhibition of CDK6 (unknown origin) | Homo sapiens | 1 | ALA5236590 | single protein format | Scientific Literature | |
| 9. | ALA5238232 | B | Inhibition of CDK7 (unknown origin) | Homo sapiens | 1 | ALA5236590 | single protein format | Scientific Literature | |
| 10. | ALA5238233 | B | Inhibition of CDK9 (unknown origin) | Homo sapiens | 1 | ALA5236590 | single protein format | Scientific Literature | |
| 11. | ALA5238234 | B | Inhibition of CDK12 (unknown origin) | Homo sapiens | 1 | ALA5236590 | single protein format | Scientific Literature | |
| 12. | ALA5238235 | B | Inhibition of human full length GSK3beta expressed in mammalian system at 1 uM by KINOMEscan analysis relative to control | Homo sapiens | 1 | ALA5236590 | assay format | Scientific Literature | |
| 13. | ALA5238236 | B | Inhibition of human partial length AMPKalphal (M1/E306) expressed in bacterial system at 1 uM by KINOMEscan analysis relative to control | Homo sapiens | 1 | ALA5236590 | assay format | Scientific Literature | |
| 14. | ALA5238237 | B | Inhibition of human partial length TAK1 (M1/Q303) expressed in mammalian system at 1 uM by KINOMEscan analysis relative to control | Homo sapiens | 1 | ALA5236590 | assay format | Scientific Literature | |
| 15. | ALA5238238 | B | Inhibition of human partial length TPKCtheta (L350/S706) expressed in bacterial system at 1 uM by KINOMEscan analysis relative to control | Homo sapiens | 1 | ALA5236590 | assay format | Scientific Literature | |
| 16. | ALA5238239 | B | Inhibition of human partial length Aurora-A (E122/K401) expressed in mammalian system at 1 uM by KINOMEscan analysis relative to control | Homo sapiens | 1 | ALA5236590 | assay format | Scientific Literature | |
| 17. | ALA5238240 | B | Inhibition of human partial length wild type DRAK1 expressed in bacterial system at 1 uM by KINOMEscan analysis relative to control | Homo sapiens | 1 | ALA5236590 | assay format | Scientific Literature | |
| 18. | ALA5238241 | B | Inhibition of human partial length wild type JAK2 (A829/G1132) expressed in mammalian system at 1 uM by KINOMEscan analysis relative to control | Homo sapiens | 1 | ALA5236590 | assay format | Scientific Literature | |
| 19. | ALA5238242 | B | Inhibition of human partial length wild type KDR (R787/P1253) expressed in mammalian system at 1 uM by KINOMEscan analysis relative to control | Homo sapiens | 1 | ALA5236590 | assay format | Scientific Literature | |
| 20. | ALA5238243 | B | Inhibition of human partial length wild type Pim-1 (M1/E291) expressed in bacterial system at 1 uM by KINOMEscan analysis relative to control | Homo sapiens | 1 | ALA5236590 | assay format | Scientific Literature |
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