| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5263166 | B | Antagonist activity at human histamine H3 receptor expressed in CHO-K1 cells assessed as inhibition of imetit-stimulation ERK1/2 phosphorylation by ELISA analysis | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
| 2. | ALA5263167 | B | Inverse agonist activity at recombinant human histamine H3 receptor expressed in CHO-K1 cells preincubated for 10 mins followed by [35S]GTPgammaS addition and measured after 60 mins by TopCount NXT based scintillation analysis | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
| 3. | ALA5263173 | B | Displacement of [3H]quinuclidinyl benzilate from Wistar rat cortex muscarinic AChR at 1 uM by liquid scintillation counting analysis relative to control | Rattus norvegicus | 18 | tissue-based format | Scientific Literature | ||
| 4. | ALA5263177 | B | Displacement of N-alpha-[methyl-3H]-methylhistamine dihydrochloride from recombinant human histamine H3 receptor expressed in CHO-K1 cells assessed as inhibition constant incubated for 30 mins by liquid scintillation analysis | Homo sapiens | 23 | cell-based format | Scientific Literature | ||
| 5. | ALA5263178 | B | Displacement of N-alpha-[methyl-3H]-methylhistamine dihydrochloride from Sprague-Dawley rat brain membrane histamine H3 receptor assessed as inhibition constant incubated for 30 mins by liquid scintillation counting analysis | Rattus norvegicus | 22 | cell membrane format | Scientific Literature |
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