| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5241960 | B | Inverse agonist activity at human GAL4-fused RORgammat LBD (262 to 507 residues) transfected in HEK293T cell assessed as maxima inhibition measured after 24 hrs by dual luciferase assay relative to control | Homo sapiens | 44 | cell-based format | Scientific Literature | ||
| 2. | ALA5241961 | B | Inverse agonist activity at human GAL4-fused FXR LBD transfected in 293T cell measured after 24 hrs by dual luciferase assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 3. | ALA5241962 | B | Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase assay | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
| 4. | ALA5241963 | B | Inverse agonist activity at human GAL4-fused LXRalpha LBD transfected in 293T cell measured after 24 hrs by dual luciferase assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 5. | ALA5241964 | B | Inverse agonist activity at human GAL4-fused RORbeta LBD transfected in 293T cell measured after 24 hrs by dual luciferase assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 6. | ALA5241965 | B | Inverse agonist activity at human GAL4-fused RORalpha LBD transfected in 293T cell measured after 24 hrs by dual luciferase assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 7. | ALA5241966 | B | Binding affinity to human RORgamma LBD (262 to 507 residues) expressed in Escherichia coli BL21(DE3) cells assessed as thermal stabilization by measuring change in melting temperature at 200 uM by thermal shift assay | Homo sapiens | 56 | cell-based format | Scientific Literature |
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