| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5261606 | B | Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | ALA5260810 | single protein format | Scientific Literature | |
| 2. | ALA5261607 | B | Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | ALA5260810 | single protein format | Scientific Literature | |
| 3. | ALA5261608 | B | Selectivity ratio of IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) to IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) | Homo sapiens | 4 | ALA5260810 | protein format | Scientific Literature | |
| 4. | ALA5261609 | B | Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | ALA5260810 | single protein format | Scientific Literature | |
| 5. | ALA5261610 | B | Selectivity ratio of IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 2 (unknown origin) to IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) | Homo sapiens | 3 | ALA5260810 | protein format | Scientific Literature | |
| 6. | ALA5261611 | B | Displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | ALA5260810 | single protein format | Scientific Literature | |
| 7. | ALA5261612 | B | Selectivity ratio of IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) to IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) | Homo sapiens | 4 | ALA5260810 | assay format | Scientific Literature | |
| 8. | ALA5261613 | B | Displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 11 | ALA5260810 | single protein format | Scientific Literature | |
| 9. | ALA5261614 | B | Binding affinity to ZsGreen fused-BRD9 (M1 to T597 residues) (unknown origin) expressed in human U2OS-C433 cells assessed as induction of protein bromodomain localization from chromatin by measuring formation of large nuclear puncta by fluorescence based assay | Homo sapiens | 10 | ALA5260810 | cell-based format | Scientific Literature | |
| 10. | ALA5261615 | B | Selectivity ratio of IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) to IC50 for displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) | Homo sapiens | 4 | ALA5260810 | assay format | Scientific Literature | |
| 11. | ALA5261633 | B | Inhibition of BRD9 in human PC-9 cells assessed as reduction in ALDH1A1 gene expression at 0.8 uM preincubated with erlotinib for 8 days followed by compound addition and measured after 24 hrs by RNA sequencing analysis | Homo sapiens | 1 | ALA5260810 | cell-based format | Scientific Literature | |
| 12. | ALA5262348 | B | Binding affinity to human partial length ATAD2A (Q981 to R1108 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 4 | ALA5260810 | assay format | Scientific Literature | |
| 13. | ALA5262349 | B | Binding affinity to human partial length ATAD2B (Q955 to R1082 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 4 | ALA5260810 | assay format | Scientific Literature | |
| 14. | ALA5262350 | B | Binding affinity to human partial length BAZ2A (M1792 to L1905 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 4 | ALA5260810 | assay format | Scientific Literature | |
| 15. | ALA5262351 | B | Binding affinity to human partial length BAZ2B (S2054 to S2168 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 4 | ALA5260810 | assay format | Scientific Literature | |
| 16. | ALA5262352 | B | Binding affinity to human partial length BRD1 (E556 to A688 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 4 | ALA5260810 | assay format | Scientific Literature | |
| 17. | ALA5262353 | B | Binding affinity to human partial length BRD2 bromodomain 1 long isoform (K71 to N194 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 4 | ALA5260810 | assay format | Scientific Literature | |
| 18. | ALA5262354 | B | Binding affinity to human partial length BRD2 bromodomain 1/2 isoform 1 (K71 to D455 residues) by BROMOscan assay | Homo sapiens | 4 | ALA5260810 | single protein format | Scientific Literature | |
| 19. | ALA5262355 | B | Binding affinity to human partial length BRD2 bromodomain 2 isoform 1 (E348 to D455 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 4 | ALA5260810 | assay format | Scientific Literature | |
| 20. | ALA5262356 | B | Binding affinity to human partial length BRD3 bromodomain 1 (P24 to E144 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 4 | ALA5260810 | assay format | Scientific Literature |
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