# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA5233078 | B | Inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) as substrate assessed as substrate hydrolysis by measuring Kinact incubated for 20 mins by colorimetric analysis | Homo sapiens | 12 | ALA5230175 | assay format | Scientific Literature | |
2. | ALA5233084 | B | Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) as substrate assessed as substrate hydrolysis by measuring KI incubated for 20 mins by colorimetric analysis | Homo sapiens | 12 | ALA5230175 | assay format | Scientific Literature | |
3. | ALA5233088 | B | Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) as substrate assessed as substrate hydrolysis by measuring Kinact/Ki ratio incubated for 20 mins by colorimetric analysis | Homo sapiens | 11 | ALA5230175 | assay format | Scientific Literature | |
4. | ALA5233090 | B | Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) as substrate assessed as substrate hydrolysis by measuring Kinact/Ki ratio by linear regression analysis | Homo sapiens | 11 | ALA5230175 | assay format | Scientific Literature | |
5. | ALA5233093 | B | Irreversible inhibition of human TG2 using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) as substrate assessed as substrate hydrolysis by measuring observed binding constant incubated for 20 mins by colorimetric assay | Homo sapiens | 4 | ALA5230175 | single protein format | Scientific Literature | |
6. | ALA5233094 | B | Irreversible inhibition of human TG1 using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) as substrate assessed as substrate hydrolysis by measuring observed binding constant incubated for 100 mins by colorimetric assay | Homo sapiens | 4 | ALA5230175 | single protein format | Scientific Literature | |
7. | ALA5233095 | B | Irreversible inhibition of human TG6 using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) as substrate assessed as substrate hydrolysis by measuring observed binding constant incubated for 60 mins by colorimetric assay | Homo sapiens | 4 | ALA5230175 | single protein format | Scientific Literature | |
8. | ALA5233096 | B | Reversible inhibition of activated human TG3 using peptidic FRET-quenched probe A101 as substrate by fluorescence based assay relative to control | Homo sapiens | 4 | ALA5230175 | single protein format | Scientific Literature | |
9. | ALA5233097 | B | Irreversible inhibition of human factor XIIIa using peptidic FRET-quenched probe A101 as substrate assessed as observed binding constant by fluorescence based assay | Homo sapiens | 3 | ALA5230175 | single protein format | Scientific Literature |