| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA832535 | B | Ex vivo effective binding dose against histamine-H1 receptor (n = 3) | Mus musculus | 8 | single protein format | Scientific Literature | ||
| 2. | ALA833040 | B | Inhibitory concentration against histamine-H1 receptor | Cavia porcellus | 20 | single protein format | Scientific Literature | ||
| 3. | ALA828053 | B | Inhibitory concentration against 5-hydroxytryptamine 2 receptor | Homo sapiens | 20 | protein format | Scientific Literature | ||
| 4. | ALA829581 | B | Binding affinity towards Alpha-1 adrenergic receptor in rat brain using [3H]prazosin as radioligand | Rattus norvegicus | 20 | tissue-based format | Scientific Literature | ||
| 5. | ALA834196 | F | Effective dose against Histamine-induced skin vascular permeability model in rat after 4 hr (n = 5) | Rattus norvegicus | 12 | organism-based format | Scientific Literature | ||
| 6. | ALA834197 | F | Effective dose against Histamine-induced skin vascular permeability model in rat after 8 hr (n = 5) | Rattus norvegicus | 7 | organism-based format | Scientific Literature | ||
| 7. | ALA914451 | B | Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum membranes | Cavia porcellus | 51 | cell membrane format | Scientific Literature | ||
| 8. | ALA914453 | B | Displacement of [3H]ketanserin from histamine H2 receptor in human cortex membranes | Homo sapiens | 51 | cell membrane format | Scientific Literature | ||
| 9. | ALA914455 | B | Displacement of [3H]prazosin from adrenergic alpha-1 receptor in rat brain membranes | Rattus norvegicus | 51 | cell membrane format | Scientific Literature | ||
| 10. | ALA914457 | F | Inhibition of increase in histamine-induced cutaneous vascular permeability in orally dosed Wistar rat model after 4 hrs | Rattus norvegicus | 36 | organism-based format | Scientific Literature | ||
| 11. | ALA914458 | F | Inhibition of increase in histamine-induced cutaneous vascular permeability in orally dosed Wistar rat model after 8 hrs | Rattus norvegicus | 18 | organism-based format | Scientific Literature | ||
| 12. | ALA914460 | F | Ex vivo displacement of [3H]mepyramine from brain histamine H1 receptor in orally dosed Swiss Albino mouse | Mus musculus | 18 | organism-based format | Scientific Literature | ||
| 13. | ALA914459 | A | Half life in Wistar rat at 1 mg/kg, iv after 8 hrs | Rattus norvegicus | 8 | organism-based format | Scientific Literature | ||
| 14. | ALA914461 | A | Volume of distribution at steady state in Wistar rat at 1 mg/kg, iv after 8 hrs | Rattus norvegicus | 8 | organism-based format | Scientific Literature | ||
| 15. | ALA914462 | A | Clearance in Wistar rat at 1 mg/kg, iv after 8 hrs | Rattus norvegicus | 8 | organism-based format | Scientific Literature | ||
| 16. | ALA914463 | F | Effect on QT interval prolongation in Dunkin-Hartley guinea pigs at 10 mg/kg, iv | Cavia porcellus | 3 | organism-based format | Scientific Literature | ||
| 17. | ALA914466 | A | Inhibition of CYP3A4 in human microsomes at 25 uM | Homo sapiens | 6 | microsome format | Scientific Literature | ||
| 18. | ALA913855 | F | Inhibition of increase in histamine-induced cutaneous vascular permeability in orally dosed Wistar rat model after 1 hrs | Rattus norvegicus | 6 | organism-based format | Scientific Literature |
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