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# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA829727 | Binding | Effective concentration against murine PPARalpha in transactivation assay | Mus musculus | 7 | ALA1145171 | single protein format | Scientific Literature | |
2. | ALA839790 | Binding | Effective concentration against human PPARalpha expressed in HepG2 cells | Homo sapiens | 16 | ALA1145171 | cell-based format | Scientific Literature | |
3. | ALA840102 | Binding | Effective concentration against human PPARgamma expressed in HepG2 cells | Homo sapiens | 16 | ALA1145171 | cell-based format | Scientific Literature | |
4. | ALA835609 | Binding | Efficacy against murine PPARalpha relative to Wy-14,643 | Mus musculus | 7 | ALA1145171 | single protein format | Scientific Literature | |
5. | ALA835610 | Binding | Efficacy against human PPARalpha expressed in HepG2 cells relative to Wy-14,643 | Homo sapiens | 16 | ALA1145171 | cell-based format | Scientific Literature | |
6. | ALA835611 | Binding | Efficacy against human PPARgamma expressed in HepG2 cells relative to rosiglitazone | Homo sapiens | 16 | ALA1145171 | cell-based format | Scientific Literature | |
7. | ALA4359317 | Binding | Inhibition of N-terminal His-tagged human PPARgamma LBD (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS assessed as S245 phosphorylation level at 10 uM by phospho gel stain method relative to control | Homo sapiens | 5 | ALA4354874 | assay format | Scientific Literature | |
8. | ALA4359318 | Binding | Inhibition of N-terminal His-tagged human PPARgamma LBD (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS assessed as reduction in S245 phosphorylation level at 10 uM incubated for 60 mins by ELISA | Homo sapiens | 2 | ALA4354874 | assay format | Scientific Literature | |
9. | ALA4359319 | Binding | Inhibition of CDK5 (unknown origin) assessed as reduction in histone H1 phosphorylation | Homo sapiens | 1 | ALA4354874 | single protein format | Scientific Literature | |
10. | ALA4359320 | Binding | Binding affinity to N-terminal His-tagged human PPARgamma LBD (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS assessed as induction of M348 cross-peak shift at 1 mol equiv by 2D 1H-15N HSQC NMR analysis | Homo sapiens | 3 | ALA4354874 | assay format | Scientific Literature | |
11. | ALA4359321 | Binding | Binding affinity to N-terminal His-tagged human PPARgamma LBD (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS assessed as induction of M348 cross-peak shift at 0.1 to 1 mol equiv by 2D 1H-15N HSQC NMR analysis | Homo sapiens | 1 | ALA4354874 | assay format | Scientific Literature | |
12. | ALA4359322 | Binding | Binding affinity to N-terminal His-tagged human PPARgamma LBD I281A mutant (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS assessed as induction of M348 cross-peak shift at 0.1 to 1 mol equiv by 2D 1H-15N HSQC NMR analysis | Homo sapiens | 1 | ALA4354874 | assay format | Scientific Literature | |
13. | ALA4359323 | Binding | Binding affinity to N-terminal His-tagged human PPARgamma LBD (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS by SPR analysis | Homo sapiens | 1 | ALA4354874 | assay format | Scientific Literature | |
14. | ALA4359324 | Binding | Binding affinity to N-terminal His-tagged human PPARgamma LBD I281A mutant (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS by SPR analysis | Homo sapiens | 1 | ALA4354874 | assay format | Scientific Literature | |
15. | ALA4359325 | Binding | Stabilization of N-terminal His-tagged human PPARgamma LBD (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS by CD spectroscopy | Homo sapiens | 1 | ALA4354874 | assay format | Scientific Literature | |
16. | ALA4359326 | Binding | Stabilization of N-terminal His-tagged human PPARgamma LBD I281A mutant (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS by CD spectroscopy | Homo sapiens | 1 | ALA4354874 | assay format | Scientific Literature | |
17. | ALA4359327 | Binding | Inhibition of N-terminal His-tagged human PPARgamma LBD I281A mutant (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS assessed as S245 phosphorylation level at 10 uM by phospho gel stain method relative to control | Homo sapiens | 3 | ALA4354874 | assay format | Scientific Literature | |
18. | ALA4359328 | Binding | Stabilization of N-terminal His-tagged human PPARgamma LBD (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS assessed as guanidine concentration to achieve 50% of folded protein incubated for 2 hrs by CD spectroscopy (Rvb = 1.69 uM) | Homo sapiens | 1 | ALA4354874 | assay format | Scientific Literature | |
19. | ALA4359329 | Binding | Inhibition of N-terminal His-tagged human PPARgamma LBD I281A mutant (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS assessed as guanidine concentration to achieve 50% of folded protein incubated for 2 hrs by CD spectroscopy (Rvb = 1.65 uM) | Homo sapiens | 1 | ALA4354874 | assay format | Scientific Literature | |
20. | ALA4359330 | Binding | Binding affinity to N-terminal His-tagged human PPARgamma LBD (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS assessed as reduction in deuterium uptake at H3 region (277 to 286 residues) by hydrogen/deuterium exchange/mass spectrometry | Homo sapiens | 1 | ALA4354874 | assay format | Scientific Literature |