| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA867061 | B | Displacement of [3H]4-OHT from ERRgamma | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 2. | ALA867062 | B | Displacement of [3H]estradiol from ERalpha | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 3. | ALA865895 | B | Selectivity for ERRgamma over ERalpha relative to 4-hydroxytamoxifen | Homo sapiens | 11 | assay format | Scientific Literature | ||
| 4. | ALA3540601 | A | Activity of human SULT1A1 expressed in escherichia coli assessed as enzyme-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation after 15 mins by Michaelis-Menten equation in presence of 20 uM PAPS | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 5. | ALA3540602 | A | Activity of human SULT1E1 expressed in escherichia coli assessed as enzyme-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation after 15 mins by Michaelis-Menten equation in presence of 20 uM PAPS | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 6. | ALA3540603 | A | Drug metabolism in human liver cytosol assessed as 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation after 15 mins by Michaelis-Menten equation in presence of 20 uM PAPS | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 7. | ALA3540604 | A | Activity of human SULT1A1 expressed in escherichia coli assessed as enzyme-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation measured per mg of protein after 15 mins by Michaelis-Menten equation in presence of 20 uM PAPS | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 8. | ALA3540605 | A | Activity of human SULT1E1 expressed in escherichia coli assessed as enzyme-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation measured per mg of protein after 15 mins by Michaelis-Menten equation in presence of 20 uM PAPS | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 9. | ALA3540882 | A | Drug metabolism in human liver cytosol assessed as 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation measured per mg of protein after 15 mins by Michaelis-Menten equation in presence of 20 uM PAPS | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA3540883 | A | Drug metabolism in human liver cytosol assessed as 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation measured per mg of protein treated with 0.1 to 30 after 15 mins by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 11. | ALA3540884 | A | Drug metabolism in human liver cytosol assessed as 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation after 15 mins by HPLC analysis in presence of 20 uM PAPS and 0.1 to 10 uM SULT1A1 inhibitor DCNP | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 12. | ALA3540885 | A | Drug metabolism in human liver cytosol assessed as SULT1A1*1/2 single nucleotide polymorphism-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 13. | ALA3540887 | A | Drug metabolism in human liver cytosol assessed as SULT1A1 copy number-1-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 14. | ALA3540888 | A | Drug metabolism in human liver cytosol assessed as SULT1A1 copy number-2-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 15. | ALA3540889 | A | Drug metabolism in human liver cytosol assessed as SULT1A1 copy number-3-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 16. | ALA3540893 | A | Drug metabolism in human liver cytosol assessed as SULT1A1 3'UTR ACG/ACG copy number-2 -mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 17. | ALA3540894 | A | Drug metabolism in human liver cytosol assessed as SULT1A1 3'UTR ACG/GTA copy number-2-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 18. | ALA3540895 | A | Drug metabolism in human liver cytosol assessed as SULT1A1 3'UTR GTA/GTA copy number-2-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 19. | ALA3540896 | A | Drug metabolism in human liver cytosol assessed as SULT1A1 3'UTR ACG/ACG copy number-3-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 20. | ALA3540897 | A | Drug metabolism in human liver cytosol assessed as SULT1A1 3'UTR ACG/GTA copy number-3-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature |
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