| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA863829 | B | Inhibition of human isolated cPLA2-alpha by vesicle assay | Homo sapiens | 14 | ALA1146074 | single protein format | Scientific Literature | |
| 2. | ALA863831 | F | Inhibition of cPLA2alpha activity assessed by A23187-induced arachidonic acid release in human platelet | Homo sapiens | 15 | ALA1146074 | assay format | Scientific Literature | |
| 3. | ALA863833 | F | Inhibition of cPLA2-alpha activity assessed by TPA-induced arachidonic acid release in human platelet | Homo sapiens | 10 | ALA1146074 | assay format | Scientific Literature | |
| 4. | ALA892787 | B | Inhibition of human platelet cPLA2-alpha assessed as arachidonic acid release by vesicle assay | Homo sapiens | 13 | ALA1147848 | assay format | Scientific Literature | |
| 5. | ALA923242 | B | Inhibition of human platelet cPLA2-alpha activity | Homo sapiens | 12 | ALA1144717 | assay format | Scientific Literature | |
| 6. | ALA923244 | A | Metabolic stability in rat liver microsomes at 20 uM after 30 mins in presence of NADPH by reverse phased HPLC relative to control | Rattus norvegicus | 12 | ALA1144717 | microsome format | Scientific Literature | |
| 7. | ALA923245 | P | Solubility in sodium phosphate buffer at pH 7.4 | 12 | ALA1144717 | small-molecule physicochemical format | Scientific Literature | ||
| 8. | ALA923246 | B | Inhibition of cPLA2-alpha in TPA-stimulated intact human platelets assessed as liberation of arachidonic acid after 60 mins | Homo sapiens | 5 | ALA1144717 | assay format | Scientific Literature | |
| 9. | ALA982355 | B | Inhibition of cPLA2 in human platelets assessed as arachidonic acid release | Homo sapiens | 9 | ALA1154396 | assay format | Scientific Literature | |
| 10. | ALA982356 | A | Metabolic stability in rat liver microsomes | Rattus norvegicus | 8 | ALA1154396 | microsome format | Scientific Literature | |
| 11. | ALA982357 | P | Thermodynamic solubility in sodium phosphate buffer at pH 7.4 | 8 | ALA1154396 | small-molecule physicochemical format | Scientific Literature | ||
| 12. | ALA1066440 | B | Inhibition of FAAH from rat brain microsomes by RP-HPLC | Rattus norvegicus | 26 | ALA1157719 | assay format | Scientific Literature | |
| 13. | ALA1066442 | B | Inhibition of cPLA2 from human platelets by RP-HPLC | Homo sapiens | 35 | ALA1157719 | assay format | Scientific Literature | |
| 14. | ALA1066445 | B | inhibition of MAGL up to 10 uM | 42 | ALA1157719 | assay format | Scientific Literature | ||
| 15. | ALA1118741 | B | Inhibition of cPLA2alpha | 2 | ALA1155440 | assay format | Scientific Literature | ||
| 16. | ALA1118742 | B | Inhibition of human platelet cPLA2alpha assessed as inhibition of arachidonic acid production after 60 mins by UV-reverse phase HPLC analysis | Homo sapiens | 30 | ALA1155440 | assay format | Scientific Literature | |
| 17. | ALA1118744 | B | Inhibition of human platelet cPLA2alpha assessed as inhibition of arachidonic acid production at 33 nM after 60 mins by UV-reverse phase HPLC analysis | Homo sapiens | 1 | ALA1155440 | assay format | Scientific Literature | |
| 18. | ALA1118745 | P | Thermodynamic solubility in sodium phosphate buffer of pH 7.4 by UV-reverse phase HPLC analysis | 34 | ALA1155440 | small-molecule physicochemical format | Scientific Literature | ||
| 19. | ALA1118746 | A | Metabolic stability in rat liver microsomes assessed as compound remaining after 30 mins by HPLC/MS analysis | Rattus norvegicus | 33 | ALA1155440 | microsome format | Scientific Literature | |
| 20. | ALA1118747 | P | Partition coefficient, log P at 5 mM by reverse phase HPLC analysis | 33 | ALA1155440 | small-molecule physicochemical format | Scientific Literature |
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