# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA615356 | B | Inhibitory activity against 20S proteosome | 2 | subcellular format | Scientific Literature | |||
2. | ALA657767 | B | Inhibitory activity against calpain at concentration up to 50 uM; No data | 1 | single protein format | Scientific Literature | |||
3. | ALA656657 | B | Inhibitory activity against cathepsin at concentration up to 50 uM; No data | 1 | single protein format | Scientific Literature | |||
4. | ALA661254 | B | Inhibitory activity against chymotrypsin at concentration up to 50 uM; No data | 1 | single protein format | Scientific Literature | |||
5. | ALA762253 | B | Inhibitory activity against papain at concentration up to 50 uM; No data | 1 | single protein format | Scientific Literature | |||
6. | ALA817280 | B | Inhibitory activity against trypsin at concentration up to 50 uM; No data | 1 | single protein format | Scientific Literature | |||
7. | ALA843997 | F | Antiproliferative activity of the compound | 8 | assay format | Scientific Literature | |||
8. | ALA852199 | F | Inhibition of the PGPH-like activity | 8 | assay format | Scientific Literature | |||
9. | ALA881728 | F | Inhibition of the chymotrypsin-like activity | 8 | assay format | Scientific Literature | |||
10. | ALA852346 | F | Inhibition of the trypsin-like activity | 8 | assay format | Scientific Literature | |||
11. | ALA861973 | B | Inhibition of chymotrypsin-like proteasome activity of human 20S proteasome | Homo sapiens | 56 | single protein format | Scientific Literature | ||
12. | ALA861974 | B | Inhibition of trypsin-like proteasome activity of human 20S proteasome | Homo sapiens | 56 | single protein format | Scientific Literature | ||
13. | ALA861975 | B | Inhibition of post glutamyl peptide hydrolase-like proteasome activity of human 20S proteasome | Homo sapiens | 56 | single protein format | Scientific Literature | ||
14. | ALA861976 | B | Inhibition of cathepsin B | Homo sapiens | 56 | single protein format | Scientific Literature | ||
15. | ALA861977 | B | Inhibition of cathepsin S | Homo sapiens | 56 | single protein format | Scientific Literature | ||
16. | ALA861978 | F | Antiproliferative activity against human PC3 cell line | Homo sapiens | 30 | cell-based format | Scientific Literature | ||
17. | ALA861979 | F | Ratio of IC50 for PC3 cells to IC50 for chymotrypsin-like proteasome activity of 20S proteasome | Homo sapiens | 23 | cell-based format | Scientific Literature | ||
18. | ALA861981 | A | Stability in human plasma after 120 mins | Homo sapiens | 30 | cell-free format | Scientific Literature | ||
19. | ALA861982 | P | Solubility in PBS at pH 7.4 | 30 | small-molecule physicochemical format | Scientific Literature | |||
20. | ALA869329 | B | Inhibition of trypsin like activity of proteasome | 6 | single protein format | Scientific Literature |