| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA864795 | B | Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranes | Rattus norvegicus | 12 | cell membrane format | Scientific Literature | ||
| 2. | ALA864797 | B | Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells | Homo sapiens | 15 | cell-based format | Scientific Literature | ||
| 3. | ALA864798 | B | Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranes | Rattus norvegicus | 12 | cell membrane format | Scientific Literature | ||
| 4. | ALA864800 | B | Displacement of [3H]MSX2 from human recombinant adenosine A2A receptor expressed in CHO cells | Homo sapiens | 15 | cell-based format | Scientific Literature | ||
| 5. | ALA864165 | B | Displacement of [3H]PSB298 from human recombinant adenosine A2B receptor expressed in CHO cells | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 6. | ALA864168 | B | Displacement of [3H]PSB11 from human recombinant adenosine A3 receptor expressed in CHO cells | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
| 7. | ALA864171 | B | Selectivity for human adenosine A2B receptor over adenosine A1 receptor | Homo sapiens | 3 | protein format | Scientific Literature | ||
| 8. | ALA864172 | B | Selectivity for human adenosine A2B receptor over adenosine A2A receptor | Homo sapiens | 3 | protein format | Scientific Literature | ||
| 9. | ALA864173 | B | Selectivity for human adenosine A2B receptor over adenosine A3 receptor | Homo sapiens | 3 | protein format | Scientific Literature | ||
| 10. | ALA864176 | B | Inhibition of [3H]PSB11 binding to human recombinant adenosine A3 receptor in CHO cells at >1 uM | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 11. | ALA2045137 | F | Antagonist activity at adenosine A2B receptor in Wistar rat ileum/jejunum segment assessed as reversal of TNBS-induced inhibition of Ach-induced contraction at 10 uM after 30 mins | Rattus norvegicus | 1 | tissue-based format | Scientific Literature | ||
| 12. | ALA2045138 | F | Antagonist activity at adenosine A2B receptor in Wistar rat ileum/jejunum segment assessed as reversal of TNBS-induced inhibition of Ach-induced contraction at 100 uM after 30 mins | Rattus norvegicus | 1 | tissue-based format | Scientific Literature | ||
| 13. | ALA2045139 | F | Antagonist activity at adenosine A2B receptor in Wistar rat ileum/jejunum segment assessed as reversal of TNBS-induced inhibition of Ach-induced contraction after 30 mins | Rattus norvegicus | 1 | tissue-based format | Scientific Literature | ||
| 14. | ALA947854 | B | Binding affinity to human adenosine A1 receptor | Homo sapiens | 10 | single protein format | Scientific Literature | ||
| 15. | ALA947855 | B | Binding affinity to human adenosine A2A receptor | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 16. | ALA947856 | B | Binding affinity to human adenosine A2B receptor | Homo sapiens | 14 | single protein format | Scientific Literature | ||
| 17. | ALA947857 | B | Binding affinity to human adenosine A3 receptor | Homo sapiens | 10 | single protein format | Scientific Literature | ||
| 18. | ALA947858 | B | Binding affinity to rat adenosine A1 receptor | Rattus norvegicus | 6 | single protein format | Scientific Literature | ||
| 19. | ALA947859 | B | Binding affinity to rat adenosine A2A receptor | Rattus norvegicus | 6 | single protein format | Scientific Literature | ||
| 20. | ALA947864 | B | Displacement of [3H]CCPA from rat brain cortex adenosine A1 receptor | Rattus norvegicus | 30 | assay format | Scientific Literature |
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