| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA685144 | F | Inhibitory concentration at which there is accumulation of UDP-[3H]-GlcNAc in the lumen of the Golgi membranes; Not determined | Oryctolagus cuniculus | 9 | ALA1129244 | cell membrane format | Scientific Literature | |
| 2. | ALA685303 | F | In vitro inhibition of UDP-[3H]-GlcNAc import into the lumen of the Golgi membranes from rabbit liver homogenate. | Oryctolagus cuniculus | 16 | ALA1129244 | tissue-based format | Scientific Literature | |
| 3. | ALA705370 | F | Inhibition of dTMP synthetase in the absence of CH2-H4 folate Lactobacillus casei | Lacticaseibacillus casei | 3 | ALA1122268 | organism-based format | Scientific Literature | |
| 4. | ALA813675 | F | Affinity towards thymidine monophosphate kinase (TMPKmt) in Mycobacterium tuberculosis | Mycobacterium tuberculosis | 4 | ALA1136204 | assay format | Scientific Literature | |
| 5. | ALA813678 | F | Kinetic parameter Vm of thymidine monophosphate kinase (TMPKmt) in Mycobacterium tuberculosis was determined | Mycobacterium tuberculosis | 4 | ALA1136204 | assay format | Scientific Literature | |
| 6. | ALA879214 | B | Compound was tested for binding affinity against Mycobacterium tuberculosis thymidine monophosphate kinase | Mycobacterium tuberculosis | 7 | ALA1135342 | single protein format | Scientific Literature | |
| 7. | ALA813680 | B | Enzyme Kinetic constant was determined in the presence of Mycobacterium tuberculosis thymidine monophosphate kinase | Mycobacterium tuberculosis | 7 | ALA1135342 | single protein format | Scientific Literature | |
| 8. | ALA815564 | B | Inhibitory activity against human thymidylate synthase with variable concentration of dUMP and fixed N5,10-CH2-H4PteGlu (200 uM) | 5 | ALA1122546 | single protein format | Scientific Literature | ||
| 9. | ALA810236 | B | The rate constant in Acetonitrile and buffered aqueous acetonitrile solution, at 30 degrees C and pH 6.8 | 3 | ALA1123535 | single protein format | Scientific Literature | ||
| 10. | ALA857842 | B | Compound was evaluated for the inhibition of dTMP synthetase with respect to dUMP. | Escherichia coli | 1 | ALA1121725 | single protein format | Scientific Literature | |
| 11. | ALA821237 | B | The compound was evaluated for the inhibition of dTMP synthetase from Lactobacillus casei | Lacticaseibacillus casei | 1 | ALA1121751 | single protein format | Scientific Literature | |
| 12. | ALA821245 | B | The apparent association constant (Ki) with dTMP synthetase enzyme from chick embryo in the absence of CH2-H4 folate was evaluated using conventional spectrophotometric assay; Active | Gallus gallus | 1 | ALA1122753 | single protein format | Scientific Literature | |
| 13. | ALA864792 | B | Inhibition of Trypanosoma cruzi dUTPase at 1 mM | Trypanosoma cruzi | 12 | ALA1137425 | single protein format | Scientific Literature | |
| 14. | ALA922718 | B | Activity at human recombinant thymidylate synthase | Homo sapiens | 2 | ALA1144764 | single protein format | Scientific Literature | |
| 15. | ALA1657145 | B | Activity at human recombinant TMPK by Michaelis-Menten equation analysis | Homo sapiens | 19 | ALA1649078 | single protein format | Scientific Literature | |
| 16. | ALA1657146 | B | Ratio of kcat/km for human recombinant TMPK by Michaelis-Menten equation analysis | Homo sapiens | 16 | ALA1649078 | single protein format | Scientific Literature | |
| 17. | ALA3255836 | B | Competitive inhibition of purified Escherichia coli thymidylate synthetase using t5-[3H]-2'-deoxyuridine 5'-phosphate as substrate after 7 mins by double reciprocal plot method | Escherichia coli | 4 | ALA3244410 | assay format | Scientific Literature | |
| 18. | ALA3255837 | B | Competitive inhibition of purified calf thymus thymidylate synthetase using 5-[3H]-2'-deoxyuridine 5'-phosphate as substrate after 7 mins by double reciprocal plot method | Bos taurus | 3 | ALA3244410 | single protein format | Scientific Literature | |
| 19. | ALA3256243 | B | Competitive inhibition of purified mouse Ehrlich ascites tumor cell thymidylate synthetase using 5-[3H]-2'-deoxyuridine 5'-phosphate as substrate after 7 mins by double reciprocal plot method | Mus musculus | 4 | ALA3244410 | single protein format | Scientific Literature | |
| 20. | ALA3284706 | B | Activity at amethopterin-resistant Lactobacillus casei thymidylate synthetase by spectrophotometric analysis in presence of CH2-H4-folate | Lacticaseibacillus casei | 1 | ALA3272104 | single protein format | Scientific Literature |
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