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| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source |
| 1. | ALA869276 | B | Displacement of [125I]NDP-MSH from human MC4R expressed in HEK293 cells | Homo sapiens | 57 | | cell-based format | Scientific Literature |
| 2. | ALA869277 | B | Inhibition of [125I]NDP-MSH binding to human MC1R expressed in HEK293 cells | Homo sapiens | 3 | | cell-based format | Scientific Literature |
| 3. | ALA869278 | B | Displacement of [125I]NDP-MSH from human MC3R expressed in HEK293 cells | Homo sapiens | 3 | | cell-based format | Scientific Literature |
| 4. | ALA869279 | B | Displacement of [125I]NDP-MSH from human MC5R expressed in HEK293 cells | Homo sapiens | 3 | | cell-based format | Scientific Literature |
| 5. | ALA869282 | F | Activity at MC4R assessed as inhibition of alpha-MSH-stimulated cAMP production | Homo sapiens | 2 | | assay format | Scientific Literature |
| 6. | ALA869280 | A | Clearance in mouse at 5 mg/kg, iv | Mus musculus | 2 | | organism-based format | Scientific Literature |
| 7. | ALA868051 | A | Volume of distribution in mouse at 5 mg/kg, iv | Mus musculus | 2 | | organism-based format | Scientific Literature |
| 8. | ALA868061 | A | Half life in mouse at 5 mg/kg, iv | Mus musculus | 2 | | organism-based format | Scientific Literature |
| 9. | ALA868057 | A | Drug level in mouse brain after 1 hr at 5 mg/kg, iv | Mus musculus | 2 | | organism-based format | Scientific Literature |
| 10. | ALA868059 | A | Drug level in mouse brain after 4 hrs at 5 mg/kg, iv | Mus musculus | 2 | | organism-based format | Scientific Literature |
| 11. | ALA868062 | A | Ratio of drug level in brain against plasma in mouse after 1 hr at 5 mg/kg, iv | Mus musculus | 2 | | organism-based format | Scientific Literature |
| 12. | ALA868060 | A | Ratio of drug level in brain against plasma in mouse after 4 hrs at 5 mg/kg, iv | Mus musculus | 2 | | organism-based format | Scientific Literature |
| 13. | ALA868055 | A | Cmax in mouse at 10 mg/kg, po | Mus musculus | 2 | | organism-based format | Scientific Literature |
| 14. | ALA868056 | A | Tmax in mouse at 10 mg/kg, po | Mus musculus | 2 | | organism-based format | Scientific Literature |
| 15. | ALA868054 | A | AUC in mouse at 10 mg/kg, po | Mus musculus | 2 | | organism-based format | Scientific Literature |
| 16. | ALA868052 | A | Bioavailability in mouse at 10 mg/kg, po | Mus musculus | 2 | | organism-based format | Scientific Literature |
| 17. | ALA868053 | P | Lipophilicity, Log D of the compound | | 2 | | small-molecule physicochemical format | Scientific Literature |
| 18. | ALA869281 | A | AUC in mouse at 5 mg/kg, iv | Mus musculus | 2 | | organism-based format | Scientific Literature |
| 19. | ALA913233 | B | Selectivity for MC4R over MC5R | Homo sapiens | 1 | | protein format | Scientific Literature |
| 20. | ALA900283 | B | Displacement of [125I]NDPMSH from human MC3R expressed in HEK293 cells | Homo sapiens | 8 | | cell-based format | Scientific Literature |