| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA909787 | B | Inhibition of Plasmodium falciparum PFT at 50 uM | Plasmodium falciparum | 42 | protein complex format | Scientific Literature | ||
| 2. | ALA910873 | B | Inhibition of Plasmodium falciparum PFT at 5 uM | Plasmodium falciparum | 34 | protein complex format | Scientific Literature | ||
| 3. | ALA910874 | F | Inhibition of Plasmodium falciparum 3D7 growth as reduced [3H]hypoxanthine incorporation | Plasmodium falciparum | 34 | organism-based format | Scientific Literature | ||
| 4. | ALA910292 | F | Inhibition of Plasmodium falciparum K1 growth as reduced [3H]hypoxanthine incorporation | Plasmodium falciparum | 34 | organism-based format | Scientific Literature | ||
| 5. | ALA910296 | A | Apparent permeability in Caco-2 cells | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 6. | ALA910297 | A | Half life in mouse liver microsome | Mus musculus | 10 | organism-based format | Scientific Literature | ||
| 7. | ALA910298 | A | Half life in rat liver microsome | Rattus norvegicus | 7 | microsome format | Scientific Literature | ||
| 8. | ALA910299 | A | AUC in mouse at 50 mg/kg, po | Mus musculus | 3 | organism-based format | Scientific Literature | ||
| 9. | ALA910300 | A | Cmax in mouse at 50 mg/kg, po | Mus musculus | 3 | organism-based format | Scientific Literature | ||
| 10. | ALA910301 | A | Half life in mouse at 50 mg/kg, po | Mus musculus | 3 | organism-based format | Scientific Literature | ||
| 11. | ALA1000383 | B | Inhibition of Plasmodium falciparum PFT | Plasmodium falciparum | 6 | assay format | Scientific Literature | ||
| 12. | ALA1000384 | B | Inhibition of Plasmodium falciparum PFT at 50 nM | Plasmodium falciparum | 39 | assay format | Scientific Literature | ||
| 13. | ALA1000385 | B | Inhibition of Plasmodium falciparum PFT at 5 nM | Plasmodium falciparum | 35 | assay format | Scientific Literature | ||
| 14. | ALA1000386 | F | Antimalarial activity in Plasmodium falciparum 3D7 infected erythrocytes as [3H]hypoxanthine uptake | Plasmodium falciparum | 35 | organism-based format | Scientific Literature | ||
| 15. | ALA1000387 | F | Antimalarial activity in Plasmodium falciparum K1 infected erythrocytes by [3H]hypoxanthine uptake | Plasmodium falciparum | 39 | organism-based format | Scientific Literature | ||
| 16. | ALA1000388 | B | Inhibition of rat PFT by scintillation proximity assay | Rattus norvegicus | 6 | assay format | Scientific Literature | ||
| 17. | ALA1000389 | B | Selectivity for Plasmodium falciparum PFT over rat PFT | 4 | assay format | Scientific Literature | |||
| 18. | ALA1260645 | B | Inhibition of human geranylgeranyltransferase-1 assessed as incorporation of [3H]GGPP into H-Ras-CVLL | Homo sapiens | 57 | protein complex format | Scientific Literature | ||
| 19. | ALA1260646 | B | Inhibition of human farnesyltransferase assessed as incorporation of [3H]FPP into H-Ras-CVLS | Homo sapiens | 57 | protein complex format | Scientific Literature | ||
| 20. | ALA1260647 | B | Selectivity ratio of IC50 for human geranylgeranyltransferase-1 to IC50 for human farnesyltransferase | Homo sapiens | 55 | assay format | Scientific Literature |
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