# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA910638 | B | Displacement of [3H]prazosin from cloned human adrenergic alpha 1A receptor expressed in CHO cells | Homo sapiens | 18 | ALA1137361 | cell-based format | Scientific Literature | |
2. | ALA910640 | B | Displacement of [3H]prazosin from cloned human adrenergic alpha 1B receptor expressed in CHO cells | Homo sapiens | 18 | ALA1137361 | cell-based format | Scientific Literature | |
3. | ALA910642 | B | Displacement of [3H]prazosin from cloned human adrenergic alpha 1D receptor expressed in CHO cells | Homo sapiens | 18 | ALA1137361 | cell-based format | Scientific Literature | |
4. | ALA910643 | B | Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampus | Rattus norvegicus | 18 | ALA1137361 | tissue-based format | Scientific Literature | |
5. | ALA910647 | B | Selectivity for human adrenergic alpha 1D receptor over human adrenergic alpha 1A receptor | Homo sapiens | 18 | ALA1137361 | protein format | Scientific Literature | |
6. | ALA912407 | B | Selectivity for human adrenergic alpha 1B receptor over human adrenergic alpha 1A receptor | Homo sapiens | 18 | ALA1137361 | protein format | Scientific Literature | |
7. | ALA912408 | B | Selectivity for 5HT1A receptor in rat hippocampus over human adrenergic alpha 1A receptor | 18 | ALA1137361 | tissue-based format | Scientific Literature | ||
8. | ALA913536 | F | Activity at adrenergic alpha 1A receptor assessed as antagonism of noradrenaline-induced contraction of Sprague-Dawley rat vas deferens | Rattus norvegicus | 12 | ALA1137361 | tissue-based format | Scientific Literature | |
9. | ALA913008 | F | Activity at adrenergic alpha 1B receptor assessed as antagonsim of phenylephrine-induced contraction of Sprague-Dawley rat spleen | Rattus norvegicus | 12 | ALA1137361 | tissue-based format | Scientific Literature | |
10. | ALA913009 | F | Activity at adrenergic alpha 1D receptor assessed as antagonism on noradrenaline-induced contraction of Sprague-Dawley rat thoracic aorta | Rattus norvegicus | 12 | ALA1137361 | tissue-based format | Scientific Literature | |
11. | ALA913010 | F | Activity at adrenergic alpha 2A receptor assessed as antagonism on noradrenaline-induced contraction of Sprague-Dawley rat vas deferens | Rattus norvegicus | 7 | ALA1137361 | tissue-based format | Scientific Literature | |
12. | ALA913011 | F | Selectivity for Sprague-Dawley rat adrenergic alpha 1B receptor over adrenergic alpha 1A receptor | Rattus norvegicus | 12 | ALA1137361 | assay format | Scientific Literature | |
13. | ALA913012 | F | Selectivity for Sprague-Dawley rat adrenergic alpha 1D receptor over adrenergic alpha 1A receptor | Rattus norvegicus | 12 | ALA1137361 | assay format | Scientific Literature | |
14. | ALA913015 | F | Inverse agonist effect on calcium-induced increase in resting tension of calcium-depleted guinea pig thoracic aorta at 10 nM | Cavia porcellus | 5 | ALA1137361 | organism-based format | Scientific Literature | |
15. | ALA2422344 | B | Selectivity ratio of Ki for human alpha-1A adrenoreceptor to Ki for 5-HT1A receptor in rat hippocampal membranes | 10 | ALA2417545 | cell membrane format | Scientific Literature | ||
16. | ALA2422543 | B | Selectivity ratio of Ki for human alpha-1A adrenoreceptor to Ki for human alpha-1B adrenoreceptor | Homo sapiens | 10 | ALA2417545 | assay format | Scientific Literature | |
17. | ALA2422544 | B | Selectivity ratio of Ki for human alpha-1A adrenoreceptor to Ki for human alpha-1D adrenoreceptor | Homo sapiens | 10 | ALA2417545 | assay format | Scientific Literature | |
18. | ALA2422545 | B | Displacement of [3H]-8-OHDPAT from 5-HT1A receptor in rat hippocampal membranes after 30 mins | Rattus norvegicus | 11 | ALA2417545 | cell membrane format | Scientific Literature | |
19. | ALA2422546 | B | Displacement of [3H]prazosin from human alpha-1D adrenoreceptor expressed in CHO cells after 30 mins | Homo sapiens | 10 | ALA2417545 | cell-based format | Scientific Literature | |
20. | ALA2422547 | B | Displacement of [3H]prazosin from human alpha-1B adrenoreceptor expressed in CHO cells after 30 mins | Homo sapiens | 10 | ALA2417545 | cell-based format | Scientific Literature |