| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA914451 | B | Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum membranes | Cavia porcellus | 51 | ALA1149258 | cell membrane format | Scientific Literature | |
| 2. | ALA914453 | B | Displacement of [3H]ketanserin from histamine H2 receptor in human cortex membranes | Homo sapiens | 51 | ALA1149258 | cell membrane format | Scientific Literature | |
| 3. | ALA914455 | B | Displacement of [3H]prazosin from adrenergic alpha-1 receptor in rat brain membranes | Rattus norvegicus | 51 | ALA1149258 | cell membrane format | Scientific Literature | |
| 4. | ALA914457 | F | Inhibition of increase in histamine-induced cutaneous vascular permeability in orally dosed Wistar rat model after 4 hrs | Rattus norvegicus | 36 | ALA1149258 | organism-based format | Scientific Literature | |
| 5. | ALA914458 | F | Inhibition of increase in histamine-induced cutaneous vascular permeability in orally dosed Wistar rat model after 8 hrs | Rattus norvegicus | 18 | ALA1149258 | organism-based format | Scientific Literature | |
| 6. | ALA914460 | F | Ex vivo displacement of [3H]mepyramine from brain histamine H1 receptor in orally dosed Swiss Albino mouse | Mus musculus | 18 | ALA1149258 | organism-based format | Scientific Literature | |
| 7. | ALA914459 | A | Half life in Wistar rat at 1 mg/kg, iv after 8 hrs | Rattus norvegicus | 8 | ALA1149258 | organism-based format | Scientific Literature | |
| 8. | ALA914461 | A | Volume of distribution at steady state in Wistar rat at 1 mg/kg, iv after 8 hrs | Rattus norvegicus | 8 | ALA1149258 | organism-based format | Scientific Literature | |
| 9. | ALA914462 | A | Clearance in Wistar rat at 1 mg/kg, iv after 8 hrs | Rattus norvegicus | 8 | ALA1149258 | organism-based format | Scientific Literature | |
| 10. | ALA914464 | F | Effect on QT interval prolongation in Dunkin-Hartley guinea pigs at 30 mg/kg, iv | Cavia porcellus | 2 | ALA1149258 | organism-based format | Scientific Literature | |
| 11. | ALA914466 | A | Inhibition of CYP3A4 in human microsomes at 25 uM | Homo sapiens | 6 | ALA1149258 | microsome format | Scientific Literature | |
| 12. | ALA913855 | F | Inhibition of increase in histamine-induced cutaneous vascular permeability in orally dosed Wistar rat model after 1 hrs | Rattus norvegicus | 6 | ALA1149258 | organism-based format | Scientific Literature |
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