# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA884939 | F | Antagonist activity against CCK2 receptor estimated from single shifts of pentagastrin concentration-effect curves in the isolated rat stomach | Rattus norvegicus | 27 | tissue-based format | Scientific Literature | ||
2. | ALA872161 | B | Concentration required to inhibit the binding of 20 pM [125I]BH-CCK-8S radioligand to guinea pig pancreas CCK1 receptor | Cavia porcellus | 31 | single protein format | Scientific Literature | ||
3. | ALA883688 | B | Concentration required to inhibit the binding of 20 pM [125I]-BH-CCK-8S radioligand to mouse cortical membrane CCK2 receptor | Mus musculus | 39 | assay format | Scientific Literature | ||
4. | ALA872181 | B | Concentration required to inhibit the binding of [125I]-BH-CCK-8S radioligand to canine gastric mucosa CCK2 receptor | Canis lupus familiaris | 5 | single protein format | Scientific Literature | ||
5. | ALA881973 | B | Percent inhibition (i.d., 3.0 mg/Kg) against dog CCK2 receptor | Canis lupus familiaris | 1 | single protein format | Scientific Literature | ||
6. | ALA881974 | B | Percent inhibition (i.v., 1.0 mg/Kg) against dog CCK2 receptor | Canis lupus familiaris | 3 | single protein format | Scientific Literature | ||
7. | ALA884376 | P | Lipophilicity was measured in octanol/buffer (pH 7.4) | 5 | small-molecule physicochemical format | Scientific Literature | |||
8. | ALA889348 | B | Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cells | Homo sapiens | 47 | cell-based format | Scientific Literature | ||
9. | ALA889350 | B | Displacement of [3H]L-364718 from human recombinant CCK1 receptor expressed in PC3 cells | Homo sapiens | 20 | cell-based format | Scientific Literature | ||
10. | ALA889352 | F | Antagonist activity at CCK2 receptor in perfused rat stomach assessed as inhibition of pentagastrin-stimulated gastric acid secretion | Rattus norvegicus | 16 | tissue-based format | Scientific Literature | ||
11. | ALA889353 | F | Displacement of [125I]BH-CCK8-8S from CCK2 receptor in canine gastric mucosa | Canis lupus familiaris | 14 | tissue-based format | Scientific Literature | ||
12. | ALA889354 | F | Inhibition of pentagastrin-stimulated gastric acid secretion in conscious gastric fistula dog at 1 mg/kg, iv | Canis lupus familiaris | 2 | organism-based format | Scientific Literature | ||
13. | ALA889355 | F | Inhibition of pentagastrin-stimulated gastric acid secretion in conscious gastric fistula dog at 0.05 mg/kg, iv | Canis lupus familiaris | 2 | organism-based format | Scientific Literature | ||
14. | ALA944976 | F | Antagonist activity at CCK2 receptor in stomach-lumen perfused immature rat | Rattus norvegicus | 21 | tissue-based format | Scientific Literature | ||
15. | ALA944977 | B | Displacement of [125I]BH-CCK-8S from CC1 receptor expressed in guinea pig pancreatic cells | Cavia porcellus | 21 | cell-based format | Scientific Literature |