| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA907546 | B | Inhibition of KDR | Homo sapiens | 34 | single protein format | Scientific Literature | ||
| 2. | ALA907547 | F | Inhibition of human KDR phosphorylation in NIH3T3 cells | Homo sapiens | 23 | cell-based format | Scientific Literature | ||
| 3. | ALA907548 | B | Selectivity for KDR over FLT1 | Homo sapiens | 2 | protein format | Scientific Literature | ||
| 4. | ALA907549 | B | Selectivity for KDR over FLT3 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 5. | ALA907550 | B | Selectivity for KDR over KIT | Homo sapiens | 2 | protein format | Scientific Literature | ||
| 6. | ALA907551 | B | Selectivity for KDR over PDGFRbeta | Homo sapiens | 2 | protein format | Scientific Literature | ||
| 7. | ALA907552 | B | Selectivity for KDR over TIE2 | Homo sapiens | 2 | protein format | Scientific Literature | ||
| 8. | ALA907553 | B | Selectivity for KDR over FGFR | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 9. | ALA907554 | B | Selectivity for KDR over cytosolic SRC | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 10. | ALA2024776 | B | Inhibition of KDR using 1 mM ATP by HTRF assay | 31 | single protein format | Scientific Literature | |||
| 11. | ALA2024777 | B | Inhibition of Aurora B using 1 mM ATP by HTRF assay | 31 | single protein format | Scientific Literature | |||
| 12. | ALA2024778 | B | Inhibition of human KDR phosphorylation expressed in mouse NIH3T3 cells | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 13. | ALA2024779 | B | Inhibition of Aurora B in human NCI-H1229 cells assessed as induction of polyploidy formation after 48 hrs by Hoechst staining-based fluorescence analysis | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 14. | ALA2024781 | F | In vivo inhibition of KDR in mouse assessed as estradiol-induced uterine edema up to 30 mg/kg, po | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 15. | ALA2024785 | A | Half life in CD1 (ICR) mouse at 3 mg/kg, iv | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 16. | ALA2024786 | A | Volume of distribution in CD1 (ICR) mouse at 3 mg/kg, iv | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 17. | ALA2024787 | A | Clearance in CD1 (ICR) mouse at 3 mg/kg, iv | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 18. | ALA2024788 | A | AUC in CD1 (ICR) mouse at 10 mg/kg, po | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 19. | ALA2024789 | A | Oral bioavailability in CD1 (ICR) mouse at 10 mg/kg | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 20. | ALA1964100 | F | PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: TOPK | 579 | assay format | PubChem BioAssays |
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