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| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source |
| 1. | ALA895698 | Binding | Displacement of [125I]ghrelin from ovine recombinant GHSR1a expressed in HEK293F cells after 6 hrs by scintillation proximity assay | Ovis aries | 38 | ALA1148824 | cell-based format | Scientific Literature |
| 2. | ALA895699 | Functional | Agonist activity at human recombinant GHSR1a expressed in HEK293F cells assessed as stimulation of [35S]GTP-gamma-S binding relative to ghrelin | Homo sapiens | 27 | ALA1148824 | cell-based format | Scientific Literature |
| 3. | ALA895700 | Functional | Antagonist activity at human recombinant GHSR1a expressed in HEK293F cells by [35S]GTP-gamma-S binding assay | Homo sapiens | 27 | ALA1148824 | cell-based format | Scientific Literature |
| 4. | ALA895702 | ADME | Cmax in Wistar rat at 3 mg/kg, po | Rattus norvegicus | 27 | ALA1148824 | organism-based format | Scientific Literature |
| 5. | ALA896830 | Binding | Displacement of [125I]DIO from 5HT2c receptor | Homo sapiens | 9 | ALA1148824 | single protein format | Scientific Literature |
| 6. | ALA896831 | Physicochemical | Aqueous solubility at pH 7.2 | | 9 | ALA1148824 | small-molecule physicochemical format | Scientific Literature |
| 7. | ALA896832 | ADME | Inhibition of CYP2D6 | | 9 | ALA1148824 | single protein format | Scientific Literature |
| 8. | ALA896833 | ADME | AUC (0-t) in Wistar rat plasma at 0.7 mg/kg, iv | Rattus norvegicus | 1 | ALA1148824 | organism-based format | Scientific Literature |
| 9. | ALA896834 | ADME | Cmax in Wistar rat plasma at 0.7 mg/kg, iv | Rattus norvegicus | 1 | ALA1148824 | organism-based format | Scientific Literature |
| 10. | ALA895697 | ADME | Half life in Wistar rat plasma at 0.7 mg/kg, iv | Rattus norvegicus | 1 | ALA1148824 | organism-based format | Scientific Literature |
| 11. | ALA896835 | ADME | Clearance in Wistar rat at 0.7 mg/kg, iv | Rattus norvegicus | 1 | ALA1148824 | organism-based format | Scientific Literature |
| 12. | ALA896836 | ADME | Volume of distribution at steady state in Wistar rat plasma at 0.7 mg/kg, iv | Rattus norvegicus | 1 | ALA1148824 | organism-based format | Scientific Literature |
| 13. | ALA896837 | ADME | AUC in Wistar rat plasma at 3 mg/kg, po | Rattus norvegicus | 2 | ALA1148824 | organism-based format | Scientific Literature |
| 14. | ALA896838 | ADME | Cmax in Wistar rat plasma at 3 mg/kg, po | Rattus norvegicus | 2 | ALA1148824 | organism-based format | Scientific Literature |
| 15. | ALA896839 | ADME | Bioavailability in Wistar rat plasma at 3 mg/kg, po | Rattus norvegicus | 3 | ALA1148824 | organism-based format | Scientific Literature |
| 16. | ALA896845 | Functional | Decrease in food intake in DIO C57BL/6 mouse at 30 mg/kg, po after 24 hrs relative to control | Mus musculus | 2 | ALA1148824 | organism-based format | Scientific Literature |
| 17. | ALA896846 | Functional | Decrease in body weight in DIO C57BL/6 mouse at 10 mg/kg, po after 9 days | Mus musculus | 1 | ALA1148824 | organism-based format | Scientific Literature |
| 18. | ALA896847 | Functional | Decrease in body weight in DIO C57BL/6 mouse at 30 mg/kg, po after 9 days | Mus musculus | 2 | ALA1148824 | organism-based format | Scientific Literature |
| 19. | ALA896848 | ADME | Cmax in po dosed DIO C57BL/6 mouse after 5 hrs | Mus musculus | 5 | ALA1148824 | organism-based format | Scientific Literature |
| 20. | ALA896849 | ADME | Drug level in po dosed DIO C57BL/6 mouse brain after 5 hrs relative to plasma concentration | Mus musculus | 5 | ALA1148824 | organism-based format | Scientific Literature |