| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA895698 | Binding | Displacement of [125I]ghrelin from ovine recombinant GHSR1a expressed in HEK293F cells after 6 hrs by scintillation proximity assay | Ovis aries | 38 | ALA1148824 | cell-based format | Scientific Literature | |
| 2. | ALA895699 | Functional | Agonist activity at human recombinant GHSR1a expressed in HEK293F cells assessed as stimulation of [35S]GTP-gamma-S binding relative to ghrelin | Homo sapiens | 27 | ALA1148824 | cell-based format | Scientific Literature | |
| 3. | ALA895700 | Functional | Antagonist activity at human recombinant GHSR1a expressed in HEK293F cells by [35S]GTP-gamma-S binding assay | Homo sapiens | 27 | ALA1148824 | cell-based format | Scientific Literature | |
| 4. | ALA895702 | ADME | Cmax in Wistar rat at 3 mg/kg, po | Rattus norvegicus | 27 | ALA1148824 | organism-based format | Scientific Literature | |
| 5. | ALA896830 | Binding | Displacement of [125I]DIO from 5HT2c receptor | Homo sapiens | 9 | ALA1148824 | single protein format | Scientific Literature | |
| 6. | ALA896831 | Physicochemical | Aqueous solubility at pH 7.2 | 9 | ALA1148824 | small-molecule physicochemical format | Scientific Literature | ||
| 7. | ALA896832 | ADME | Inhibition of CYP2D6 | 9 | ALA1148824 | single protein format | Scientific Literature |
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