| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA931094 | F | Antagonist activity at dopamine D3 receptor by GTPgammaS binding assay | 36 | assay format | Scientific Literature | |||
| 2. | ALA931096 | F | Antagonist activity at dopamine D2 receptor by GTPgammaS binding assay | 36 | assay format | Scientific Literature | |||
| 3. | ALA931103 | F | Antagonist activity at histamine H1 receptor by FLIPR assay | 36 | assay format | Scientific Literature | |||
| 4. | ALA931097 | B | Inhibition of human ERG | Homo sapiens | 36 | single protein format | Scientific Literature | ||
| 5. | ALA931098 | B | Selectivity for dopamine D3 receptor over dopamine D2 receptor | 36 | assay format | Scientific Literature | |||
| 6. | ALA931104 | B | Selectivity for dopamine D3 receptor over histamine H1 receptor | 36 | assay format | Scientific Literature | |||
| 7. | ALA931105 | B | Selectivity for dopamine D3 receptor over human ERG | 36 | assay format | Scientific Literature | |||
| 8. | ALA895461 | F | Displacement of [35S]GTP-gamma-S from human cloned dopamine D3 receptor expressed in CHO cells after 30 mins | Homo sapiens | 42 | cell-based format | Scientific Literature | ||
| 9. | ALA895462 | F | Displacement of [35S]GTP-gamma-S from human cloned dopamine D2 receptor expressed in CHO cells after 30 mins | Homo sapiens | 42 | cell-based format | Scientific Literature | ||
| 10. | ALA895463 | F | Binding affinity to human histamine H1 receptor expressed in CHO cells by FLIPR assay | Homo sapiens | 42 | cell-based format | Scientific Literature | ||
| 11. | ALA895464 | B | Displacement of [3H]dofetilide from hERG expressed in CHO cells | Homo sapiens | 42 | cell-based format | Scientific Literature | ||
| 12. | ALA895468 | A | Volume of distribution in Sprague-Dawley rat | Rattus norvegicus | 4 | organism-based format | Scientific Literature | ||
| 13. | ALA895471 | A | Inhibition of human cytochrome P450 at <10 uM | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA895472 | A | Intrinsic clearance in human liver microsome | Homo sapiens | 3 | microsome format | Scientific Literature | ||
| 15. | ALA895473 | A | Blood clearance in Sprague-Dawley rat at 20 mg/kg after 30 mins | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 16. | ALA895474 | A | Bioavailability in Sprague-Dawley rat at 20 mg/kg after 30 mins | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 17. | ALA895475 | A | Volume of distribution in Sprague-Dawley rat at 20 mg/kg after 30 mins | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 18. | ALA895476 | A | Half life in Sprague-Dawley rat at 20 mg/kg after 30 mins | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 19. | ALA895477 | A | Ratio of drug level in blood to brain in Sprague-Dawley rat at 20 mg/kg after 30 mins | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 20. | ALA895478 | B | Binding affinity to hERG expressed in CHO cells by patch clamp assay | Homo sapiens | 2 | cell-based format | Scientific Literature |
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