| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA633649 | A | Delta logD (logD6.5 - logD7.4) | 111 | ALA1133765 | assay format | Scientific Literature | ||
| 2. | ALA634283 | P | Partition coefficient (logD6.5) | 114 | ALA1133765 | small-molecule physicochemical format | Scientific Literature | ||
| 3. | ALA645153 | P | Ionization constant (pKa) | 204 | ALA1133765 | small-molecule physicochemical format | Scientific Literature | ||
| 4. | ALA633098 | A | Oral bioavailability in human | Homo sapiens | 184 | ALA1133765 | organism-based format | Scientific Literature | |
| 5. | ALA719738 | F | Effective dose required to produce analgesic action in mice after peroral administration | Mus musculus | 24 | ALA1122844 | organism-based format | Scientific Literature | |
| 6. | ALA735323 | F | Analgesic agonist activity in acetic acid induced mouse writhing assay, subcutaneous administration | Mus musculus | 28 | ALA1121639 | organism-based format | Scientific Literature | |
| 7. | ALA754959 | B | Binding affinity against opioid receptor mu using [3H]-DAMGO as radioligand. | 34 | ALA1125499 | single protein format | Scientific Literature | ||
| 8. | ALA763607 | B | Binding affinity against PCP receptor using [3H]TCP as radioligand. | 34 | ALA1125499 | assay format | Scientific Literature | ||
| 9. | ALA763608 | B | Ratio of binding affinities of pcp receptor(ki(nM)) to sigma opioid receptor(ki(nM)) | 34 | ALA1125499 | assay format | Scientific Literature | ||
| 10. | ALA781188 | F | Narcotic antagonist activity against an ED80 of morphine in the modified rat tail-flick assay | Rattus norvegicus | 16 | ALA1121639 | organism-based format | Scientific Literature | |
| 11. | ALA805774 | B | Binding affinity against sigma opioid receptor using [3H]pentazocine as radioligand. | 24 | ALA1125499 | assay format | Scientific Literature | ||
| 12. | ALA809834 | B | Affinity against Sigma opioid receptor type 1 using [3H](+)-pentazocine in guinea pig brain membranes | Cavia porcellus | 18 | ALA1132466 | cell membrane format | Scientific Literature | |
| 13. | ALA808280 | B | Affinity against Sigma opioid receptor type 2 using [3H]- DTG in rat liver membranes | Rattus norvegicus | 18 | ALA1132466 | cell membrane format | Scientific Literature | |
| 14. | ALA809882 | B | Tested for binding affinity against sigma receptors | Cavia porcellus | 3 | ALA1127639 | single protein format | Scientific Literature | |
| 15. | ALA809040 | B | Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranes | 25 | ALA1133659 | cell membrane format | Scientific Literature | ||
| 16. | ALA808205 | B | Binding affinity measured on Sigma receptor type 1 from guinea pig brain membranes using [3H]pentazocine as radioligand. | Cavia porcellus | 20 | ALA1128493 | assay format | Scientific Literature | |
| 17. | ALA808206 | B | Binding affinity was measured on Sigma receptor type 1 using [3H]- pentazocine as radioligand | Cavia porcellus | 3 | ALA1128494 | single protein format | Scientific Literature | |
| 18. | ALA809515 | B | Compound was evaluated for the binding affinity towards Sigma receptor type 1 using radioligand ([3H]-(+)- Pentazocine) binding assay. | 41 | ALA1128387 | single protein format | Scientific Literature | ||
| 19. | ALA809516 | B | Binding affinity towards sigma receptor binding site 1 using [3H](+)-pentazocine | 33 | ALA1128738 | single protein format | Scientific Literature | ||
| 20. | ALA809517 | B | Ratio of the binding affinities against Sigma receptor type 1 and Sigma receptor type 2 | 41 | ALA1128387 | single protein format | Scientific Literature |
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