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# Aladdin ID Assay Type Description Organism Compounds Reference BAO Format Source 1. ALA720015 F Percent inhibition of convulsions in audiogenic DBA/2 mice at dose 20 mg/kg Mus musculus 6 ALA1131053 organism-based format Scientific Literature 2. ALA780515 F Inhibitory effect against veratridine-induced glutamate release from rat brain slices Rattus norvegicus 33 ALA1135973 assay format Scientific Literature 3. ALA787012 F Percent inhibition of veratridine-induced glutamate release in rat brain slices at 10000 nmol/L; ND is No Data. Rattus norvegicus 4 ALA1135973 tissue-based format Scientific Literature 4. ALA789319 F Neuroprotective activity was determined in the rat middle cerebral artery occlusion (MCAO) model of focal stroke Rattus norvegicus 13 ALA1134457 organism-based format Scientific Literature 5. ALA806327 B In vitro inhibition of [14C]- guanidinium influx in Chinese hamster ovary (CHO) cells expressing rat brain sodium channel type IIA (CNaIIA-1) Rattus norvegicus 12 ALA1131053 cell-based format Scientific Literature 6. ALA818548 B Inhibition of [3H]BTX binding to cardiac voltage-gated sodium channel Rattus norvegicus 15 ALA1134457 assay format Scientific Literature 7. ALA845816 B Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomes Rattus norvegicus 33 ALA1135973 subcellular format Scientific Literature 8. ALA844979 B Displacement of [3H]-MK-801 from rat cerebral cortex glutamate NMDA receptor; ND is No Data. Rattus norvegicus 3 ALA1135973 tissue-based format Scientific Literature 9. ALA1027763 A Volume of distribution at steady state in human Homo sapiens 5 ALA1158480 organism-based format Scientific Literature 10. ALA1028540 A Volume of distribution at steady state in human administered three way cross over study in 11, 10 and 12 healthy subjects at 5, 10, 15 mg dose respectively as 1 hr infusion Homo sapiens 1 ALA1158480 organism-based format Scientific Literature 11. ALA1028541 A Clearance in human administered three way cross over study in 11, 10 and 12 healthy subjects at 5, 10, 15 mg dose respectively as 1 hr infusion Homo sapiens 1 ALA1158480 organism-based format Scientific Literature 12. ALA1028542 A Mean residence time in human administered three way cross over study in 11, 10 and 12 healthy subjects at 5, 10, 15 mg dose respectively as 1 hr infusion Homo sapiens 1 ALA1158480 organism-based format Scientific Literature 13. ALA1028543 A Half life in human administered three way cross over study in 11, 10 and 12 healthy subjects at 5, 10, 15 mg dose respectively as 1 hr infusion Homo sapiens 1 ALA1158480 organism-based format Scientific Literature 14. ALA1028544 A Volume of distribution at steady state in human given 31 administration across 6 doses 2.5 to 25 mg administered 30 mins infusion each dose separated by 13 days Homo sapiens 1 ALA1158480 organism-based format Scientific Literature 15. ALA1028545 A Clearance in human given 31 administration across 6 doses 2.5 to 25 mg administered 30 mins infusion each dose separated by 13 days Homo sapiens 1 ALA1158480 organism-based format Scientific Literature 16. ALA1028546 A Mean residence time in human given 31 administration across 6 doses 2.5 to 25 mg administered 30 mins infusion each dose separated by 13 days Homo sapiens 1 ALA1158480 organism-based format Scientific Literature 17. ALA1028547 A Half life in human given 31 administration across 6 doses 2.5 to 25 mg administered 30 mins infusion each dose separated by 13 days Homo sapiens 1 ALA1158480 organism-based format Scientific Literature 18. ALA2416952 F Cytotoxicity against human A2780 cells after 72 hrs by MTT assay Homo sapiens 3 ALA2413002 cell-based format Scientific Literature 19. ALA2416953 F Cytotoxicity against human A549 cells after 72 hrs by MTT assay Homo sapiens 3 ALA2413002 cell-based format Scientific Literature 20. ALA2416954 F Antiproliferative activity against human A2780 cells at 0.005 uM after 72 hrs by MTT assay Homo sapiens 1 ALA2413002 cell-based format Scientific Literature