| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA895641 | B | Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CHOK1 cells | Homo sapiens | 53 | cell-based format | Scientific Literature | ||
| 2. | ALA895642 | B | Displacement of [125I]NDP-alphaMSH from human melanocortin 1 receptor expressed in CHOK1 cells | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 3. | ALA895643 | B | Displacement of [125I]NDP-alphaMSH from human melanocortin 3 receptor expressed in CHOK1 cells | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 4. | ALA895644 | B | Displacement of [125I]NDP-alphaMSH from human melanocortin 5 receptor expressed in CHOK1 cells | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 5. | ALA895645 | F | Antagonist activity at human melanocortin 4 receptor expressed in CHOK1 cells assessed as inhibition of NDP-alpha-MSH-stimulated cAMP production | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 6. | ALA895646 | A | Half life in Sprague-Dawley rat at 4.5 umol/kg, iv | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 7. | ALA896762 | A | Ratio of drug level in brain to blood in Sprague-Dawley rat at 4.5 umol/kg, iv | Rattus norvegicus | 1 | tissue-based format | Scientific Literature | ||
| 8. | ALA896763 | B | Selectivity for human MC4R over human MC3R | Homo sapiens | 4 | protein format | Scientific Literature | ||
| 9. | ALA896764 | F | Agonist activity at human melanocortin 4 receptor expressed in CHOK1 cells assessed as stimulation of cAMP production at 10 uM | Homo sapiens | 4 | cell-based format | Scientific Literature |
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