| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA899759 | B | Binding affinity at human MC4R | Homo sapiens | 42 | single protein format | Scientific Literature | ||
| 2. | ALA899757 | A | Inhibition of microsomal CYP3A4 | 42 | assay format | Scientific Literature | |||
| 3. | ALA899758 | F | Antagonist activity at human MC4R expressed in HEK293 cells by cAMP accumulation assay | Homo sapiens | 15 | cell-based format | Scientific Literature | ||
| 4. | ALA899754 | B | Binding affinity at human MC1R at 10 uM | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 5. | ALA899755 | B | Binding affinity at human MC3R | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 6. | ALA899753 | B | Binding affinity at mouse MC3R | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 7. | ALA899752 | B | Binding affinity at rat MC3R | Rattus norvegicus | 1 | single protein format | Scientific Literature | ||
| 8. | ALA899750 | B | Binding affinity at mouse MC4R | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 9. | ALA899760 | B | Binding affinity at rat MC4R | Rattus norvegicus | 1 | single protein format | Scientific Literature | ||
| 10. | ALA899761 | B | Binding affinity at human MC5R | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 11. | ALA899762 | A | Plasma clearance in mouse at 5 mg/kg, iv | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 12. | ALA899763 | A | Volume of distribution in mouse at 5 mg/kg, iv | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 13. | ALA899764 | A | Half life in mouse at 5 mg/kg, iv | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 14. | ALA899765 | A | AUC in mouse at 5 mg/kg, iv | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 15. | ALA899766 | A | Drug level in mouse brain at 5 mg/kg, iv after 1 hr | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 16. | ALA899767 | A | Drug level in mouse brain at 5 mg/kg, iv after 4 hrs | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 17. | ALA899768 | A | Ratio of drug level in brain to plasma in rat at 5 mg/kg, iv after 1 hr | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 18. | ALA899769 | A | Cmax in mouse at 10 mg/kg, po after 2 hrs | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 19. | ALA899770 | A | Tmax in mouse at 10 mg/kg, po | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 20. | ALA899771 | A | AUC in mouse at 10 mg/kg, po | Mus musculus | 1 | organism-based format | Scientific Literature |
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