| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA624570 | A | Oral bioavailability in human | Homo sapiens | 1 | organism-based format | Scientific Literature | ||
| 2. | ALA623353 | A | Oral bioavailability administered in solution in rats | Canis lupus familiaris | 1 | organism-based format | Scientific Literature | ||
| 3. | ALA621342 | A | Area under curve was measured by using concentration Vs time | 17 | assay format | Scientific Literature | |||
| 4. | ALA626164 | A | Area under curve gives the effective duration for the angiotensin II antagonist effect. | 13 | assay format | Scientific Literature | |||
| 5. | ALA628702 | A | Oral bioavailability in rat | Rattus norvegicus | 3 | organism-based format | Scientific Literature | ||
| 6. | ALA633713 | P | Partition coefficient (logP) | 8 | small-molecule physicochemical format | Scientific Literature | |||
| 7. | ALA647289 | B | Displacement of [1251][Sar1,IIe8]AII from rabbit aorta Angiotensin II receptor, type 1 | Oryctolagus cuniculus | 13 | tissue-based format | Scientific Literature | ||
| 8. | ALA648938 | F | Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic rings | Oryctolagus cuniculus | 10 | assay format | Scientific Literature | ||
| 9. | ALA649713 | F | In vitro antagonism of Angiotensin II receptor, type 1 in isolated rabbit thoracic aorta | Oryctolagus cuniculus | 9 | tissue-based format | Scientific Literature | ||
| 10. | ALA647927 | B | Compound was evaluated for in vitro potency against angiotensin II receptor, type 1 in isolated rabbit aorta; value ranges from 8.27-8.70 | Oryctolagus cuniculus | 1 | single protein format | Scientific Literature | ||
| 11. | ALA645253 | B | Potency to antagonize the ability of angiotensin II to contract rabbit aorta | Oryctolagus cuniculus | 100 | tissue-based format | Scientific Literature | ||
| 12. | ALA645254 | B | pA2 value determined in vitro against angiotensin II receptor, type 1 using rabbit aortic rings | Oryctolagus cuniculus | 40 | single protein format | Scientific Literature | ||
| 13. | ALA646327 | F | Angiotensin II receptor, type 1 antagonist activity in rabbit isolated thoracic aorta | Oryctolagus cuniculus | 15 | tissue-based format | Scientific Literature | ||
| 14. | ALA644579 | B | Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]angiotensin II binding to rat uterine membrane. | 15 | assay format | Scientific Literature | |||
| 15. | ALA644580 | B | Binding affinity against angiotensin II receptor type 1 (AT1) from rat liver. | 37 | assay format | Scientific Literature | |||
| 16. | ALA644582 | B | Binding affinity for Angiotensin II receptor, type 1 measured by ability to displace [125I]- A II from its specific binding site in rat liver membrane | 52 | cell membrane format | Scientific Literature | |||
| 17. | ALA648960 | B | Concentration required to inhibit binding of radioligand [125I]AII to angiotensin II receptor, type 1 in rat adrenal glomerulosa tissue | 7 | assay format | Scientific Literature | |||
| 18. | ALA648961 | B | Binding affinity for rat angiotensin II receptor, type 1 | 42 | single protein format | Scientific Literature | |||
| 19. | ALA648963 | B | Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparation | 42 | cell membrane format | Scientific Literature | |||
| 20. | ALA648755 | F | In vitro antagonistic activity by displacement of [125I]-Sar1-Ile8-A II at the rat adrenal cortical aorta Angiotensin II receptor, type 1 | 1 | tissue-based format | Scientific Literature |
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