| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA885775 | B | Displacement of [3H]N-alpha-methylhistamine from human cloned histamine H3 receptor expressed in C6 cells | Homo sapiens | 24 | cell-based format | Scientific Literature | ||
| 2. | ALA885776 | B | Displacement of [3H]N-alpha-methylhistamine from histamine H3 receptor in rat cortical membranes | Rattus norvegicus | 22 | cell membrane format | Scientific Literature | ||
| 3. | ALA885777 | A | Half life in rat at 1 mg/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 4. | ALA885778 | A | Volume of distribution in rat at terminal phase at 1 mg/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 5. | ALA885779 | A | AUC (0 to infinity) in rat at 1 mg/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 6. | ALA885780 | A | Clearance in rat brain at 1 mg/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 7. | ALA885781 | A | Cmax in rat at 1 mg/kg, po | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 8. | ALA885782 | A | Half life in rat at 1 mg/kg, po | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 9. | ALA885783 | A | AUC (0 to infinity) in rat at 1 mg/kg, po | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 10. | ALA885784 | A | Oral bioavailability in rat at 1 mg/kg | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 11. | ALA885785 | A | Ratio of drug level in brain to plasma in rat at 5 mg/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 12. | ALA885786 | B | Selectivity for human histamine H3 receptor over human histamine H1 receptor | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA885787 | B | Selectivity for human histamine H3 receptor over human histamine H2 receptor | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA885788 | B | Selectivity for human histamine H3 receptor over human histamine H4 receptor | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA2154938 | B | Binding affinity to rat cortical histamine H3 receptor | Rattus norvegicus | 11 | single protein format | Scientific Literature | ||
| 16. | ALA2154939 | B | Binding affinity to human histamine H3 receptor | Homo sapiens | 20 | single protein format | Scientific Literature | ||
| 17. | ALA2154943 | A | Oral bioavailability in rat | Rattus norvegicus | 4 | organism-based format | Scientific Literature | ||
| 18. | ALA2154944 | A | Half life in rat | Rattus norvegicus | 5 | organism-based format | Scientific Literature |
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