| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA751847 | B | Inhibition of [3H]-nicotinic acid (20 nM) binding to nicotinic acid receptor in rat spleen membrane. | Rattus norvegicus | 20 | cell membrane format | Scientific Literature | ||
| 2. | ALA784063 | F | G protein activation was measured by stimulation of [35S]GTP gamma-S binding to rat adipocyte membranes | Rattus norvegicus | 9 | organism-based format | Scientific Literature | ||
| 3. | ALA787015 | F | Potency required for stimulation of [35S]-GTP gamma-S binding to rat spleen was determined; Not determined | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 4. | ALA787016 | F | Relative intrinsic activity in stimulation of [35S]GTP gamma-S binding to rat spleen was determined; Not determined | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 5. | ALA794202 | F | Relative intrinsic activity in stimulation of [35S]GTP gamma-S binding to rat adipocyte was determined | Rattus norvegicus | 9 | organism-based format | Scientific Literature | ||
| 6. | ALA924060 | F | Agonist activity at human cloned GPR109a receptor by forskolin-stimulated cAMP production test | Homo sapiens | 41 | assay format | Scientific Literature | ||
| 7. | ALA921658 | F | Agonist activity at GPR109A receptor expressed in CHOK1 cells assessed as inhibition of forskolin-induced intracellular cAMP production by Flashplate assay | 7 | cell-based format | Scientific Literature | |||
| 8. | ALA921659 | F | Agonist activity at GPR109A receptor expressed in CHOK1 cells assessed as inhibition of forskolin-induced intracellular cAMP production by Flashplate assay relative to nicotinic acid | 7 | cell-based format | Scientific Literature | |||
| 9. | ALA921660 | F | Inhibition of isoproterenol-induced lipolysis in human subcutaneous adipocytes after 5 hrs | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 10. | ALA921661 | F | Reduction of free fatty acid level in ip dosed C57/BL6 mouse plasma after 10 mins | Mus musculus | 6 | organism-based format | Scientific Literature | ||
| 11. | ALA921662 | F | Reduction of free fatty acid level in po dosed Sprague-Dawley rat plasma | Rattus norvegicus | 6 | organism-based format | Scientific Literature | ||
| 12. | ALA921663 | F | Reduction of free fatty acid level in po dosed Sprague-Dawley rat plasma relative to baseline | Rattus norvegicus | 6 | organism-based format | Scientific Literature | ||
| 13. | ALA921664 | A | Induction of flushing response in ip dosed C57/BL6 mouse | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 14. | ALA921665 | F | Inhibition of nicotinic acid induced flushing response in ip dosed C57/BL6 mouse | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 15. | ALA921666 | B | Activation of GPR109A receptor in CHOK1 cells assessed as ERK1/2 MAP kinase activation by ELISA | 4 | cell-based format | Scientific Literature | |||
| 16. | ALA933836 | B | Induction of internalization of epitope-tagged GPR109A receptor expressed in COS7 cells after 30 mins | 2 | cell-based format | Scientific Literature | |||
| 17. | ALA933837 | B | Induction of internalization of epitope-tagged GPR109A receptor expressed in COS7 cells at 10 uM after 30 mins | 4 | cell-based format | Scientific Literature |
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