| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3436220 | Functional | Inhibition of L-type calcium channel measured using whole-cell patch clamp in guinea pig ventricular myocytes | Cavia porcellus | 1 | ALA3436046 | cell-based format | Scientific Literature | |
| 2. | ALA3436221 | Functional | Inhibition of L-type calcium channel measured using 2-electrode voltage-clamp in Xenopus oocyte heterologically expressing alpha-1C subunit | Xenopus | 1 | ALA3436046 | cell-based format | Scientific Literature | |
| 3. | ALA3436222 | Functional | Inhibition of L-type calcium channel measured using 2-electrode voltage-clamp in Xenopus oocyte heterologically expressing alpha-1C subunit | Xenopus | 1 | ALA3436046 | cell-based format | Scientific Literature | |
| 4. | ALA3534882 | ADME | Time dependent inhibition of CYP1A2 (unknown origin) at 100 uM by LC/MS system | Homo sapiens | 42 | ALA3526118 | single protein format | Scientific Literature | |
| 5. | ALA3534885 | ADME | Time dependent inhibition of CYP2C19 in human liver microsomes at 100 uM by LC/MS system | Homo sapiens | 38 | ALA3526118 | assay format | Scientific Literature | |
| 6. | ALA3534886 | ADME | Time dependent inhibition of CYP2D6 (unknown origin) at 100 uM by LC/MS system | Homo sapiens | 37 | ALA3526118 | single protein format | Scientific Literature | |
| 7. | ALA3534887 | ADME | Time dependent inhibition of CYP3A4 (unknown origin) at 100 uM by LC/MS system | Homo sapiens | 35 | ALA3526118 | single protein format | Scientific Literature | |
| 8. | ALA3534888 | ADME | Covalent binding in human liver microsomes measured per mg of protein using radiolabelled compound at 10 uM after 1 hr incubation by liquid scintillation counting | Homo sapiens | 42 | ALA3526118 | assay format | Scientific Literature | |
| 9. | ALA3534889 | ADME | Metabolic activation in human liver microsomes assessed as [3H]GSH adduct formation rate measured per mg of protein at 100 uM by [3H]GSH trapping assay | Homo sapiens | 42 | ALA3526118 | assay format | Scientific Literature | |
| 10. | ALA3534890 | ADME | Time dependent inhibition of CYP2C8 (unknown origin) at 100 uM by LC/MS system | Homo sapiens | 34 | ALA3526118 | single protein format | Scientific Literature | |
| 11. | ALA3534891 | ADME | Time dependent inhibition of CYP3A4 (unknown origin) at 10 uM by LC/MS system | Homo sapiens | 6 | ALA3526118 | single protein format | Scientific Literature | |
| 12. | ALA3534895 | ADME | Time dependent inhibition of CYP2C9 (unknown origin) at 30 uM by LC/MS system | Homo sapiens | 3 | ALA3526118 | single protein format | Scientific Literature | |
| 13. | ALA3534902 | ADME | Time dependent inhibition of CYP2D6 (unknown origin) at 30 uM by LC/MS system | Homo sapiens | 2 | ALA3526118 | single protein format | Scientific Literature | |
| 14. | ALA3534905 | ADME | Intrinsic clearance for reactive metabolites formation per mg of protein in human liver microsomes based on [3H]GSH adduct formation rate at 100 uM by [3H]GSH trapping assay | Homo sapiens | 42 | ALA3526118 | assay format | Scientific Literature | |
| 15. | ALA3534906 | ADME | Intrinsic clearance for reactive metabolites formation per mg of protein based on cytochrome P450 (unknown origin) inactivation rate by TDI assay | Homo sapiens | 42 | ALA3526118 | assay format | Scientific Literature | |
| 16. | ALA3534907 | ADME | Intrinsic clearance for reactive metabolites formation assessed as summation of [3H]GSH adduct formation rate-based reactive metabolites formation and cytochrome P450 (unknown origin) inactivation rate-based reactive metabolites formation | Homo sapiens | 42 | ALA3526118 | assay format | Scientific Literature | |
| 17. | ALA3532420 | ADME | Time dependent inhibition of CYP2B6 (unknown origin) at 3 uM by LC/MS system | Homo sapiens | 1 | ALA3526118 | single protein format | Scientific Literature | |
| 18. | ALA3561978 | Functional | PubChem BioAssay. nuclear beta catenin stimulation in WNT3A conditioned C2C12 cells-IC50. (Class of assay: confirmatory) | 97 | ALA1201862 | cell-based format | PubChem BioAssays | ||
| 19. | ALA3562024 | Functional | PubChem BioAssay. VEGF stimulated ADSC/ECFC co-culture nuclear area decrease (viability)-IC50. (Class of assay: confirmatory) | 369 | ALA1201862 | assay format | PubChem BioAssays | ||
| 20. | ALA3562043 | Functional | PubChem BioAssay. VEGF stimulated ADSC/ECFC co-culture CD31-stained tube area decrease-IC50. (Class of assay: confirmatory) | 368 | ALA1201862 | assay format | PubChem BioAssays |
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