| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1805697 | Binding | Inhibition of PDE4A | 19 | ALA1799977 | single protein format | Scientific Literature | ||
| 2. | ALA1805698 | Binding | Inhibition of PDE4B | 19 | ALA1799977 | single protein format | Scientific Literature | ||
| 3. | ALA1805699 | Binding | Inhibition of PDE4D | 19 | ALA1799977 | single protein format | Scientific Literature | ||
| 4. | ALA1805700 | Binding | Inhibition of PDE4 activity in human whole blood assessed as inhibition of LPS-induced TNF-alpha release | Homo sapiens | 19 | ALA1799977 | protein format | Scientific Literature | |
| 5. | ALA1805702 | ADME | Competitive inhibition of CYP2C9 | 3 | ALA1799977 | single protein format | Scientific Literature | ||
| 6. | ALA1804291 | Binding | Ratio IC50 for PDE4 activity in human whole blood to IC50 for PDE4 | 19 | ALA1799977 | tissue-based format | Scientific Literature | ||
| 7. | ALA945012 | Functional | Inhibition of LPS-stimulated TNFalpha release in squirrel monkey whole blood | Saimiri sciureus | 3 | ALA1141472 | tissue-based format | Scientific Literature | |
| 8. | ALA945013 | ADME | Inhibition of CYP2C9 | 17 | ALA1141472 | single protein format | Scientific Literature | ||
| 9. | ALA945014 | Binding | Inhibition of PDE4 expressed in SF9 cells | 27 | ALA1141472 | cell-based format | Scientific Literature | ||
| 10. | ALA945015 | Functional | Inhibition of LPS-stimulated TNFalpha release in human whole blood | Homo sapiens | 27 | ALA1141472 | tissue-based format | Scientific Literature | |
| 11. | ALA945016 | ADME | Oral bioavailability in rat | Rattus norvegicus | 14 | ALA1141472 | organism-based format | Scientific Literature | |
| 12. | ALA945017 | ADME | Half life in rat | Rattus norvegicus | 14 | ALA1141472 | organism-based format | Scientific Literature | |
| 13. | ALA945019 | ADME | Cmax in squirrel monkey at 10 mg/kg | Saimiri sciureus | 2 | ALA1141472 | organism-based format | Scientific Literature | |
| 14. | ALA945962 | ADME | Therapeutic index, ratio of plasma concentration causing emesis to IC50 for inhibition of LPS-stimulated TNFalpha release in squirrel monkey whole blood | Saimiri sciureus | 3 | ALA1141472 | cell-free format | Scientific Literature | |
| 15. | ALA945963 | Functional | Inhibition of ovalbumin-induced bronchoconstriction in guinea pig at 30 ug/kg, ip | Cavia porcellus | 2 | ALA1141472 | organism-based format | Scientific Literature |
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