# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA650284 | Binding | The percent inhibition of [3H]diazepam binding to the benzodiazepine receptor of rat brain elicited by 100 uM of compound | 28 | ALA1124455 | assay format | Scientific Literature | ||
2. | ALA758627 | Binding | Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding site | 53 | ALA1124860 | protein format | Scientific Literature | ||
3. | ALA758630 | Binding | Binding affinity (Ki) against human phosphatidylinositol 4-kinase | 51 | ALA1124860 | protein format | Scientific Literature | ||
4. | ALA939343 | Binding | Inhibition of p34cdc2/cyclin B | 3 | ALA1145498 | assay format | Scientific Literature | ||
5. | ALA939344 | Functional | Cell cycle arrest in human HeLa cells assessed as accumulation at S phase | Homo sapiens | 2 | ALA1145498 | cell-based format | Scientific Literature | |
6. | ALA3301363 | Physicochemical | ASTRAZENECA: Octan-1-ol/water (pH7.4) distribution coefficent measured by a shake flask method described in J. Biomol. Screen. 2011, 16, 348-355. Experimental range -1.5 to 4.5 | 4,197 | ALA3301361 | small-molecule physicochemical format | AstraZeneca Deposited Data | ||
7. | ALA1648129 | Binding | Inhibition of ASK1 assessed as phosphorylated fluorescent peptide at 10 uM by mobility shift assay | 21 | ALA1641590 | single protein format | Scientific Literature | ||
8. | ALA1963690 | Functional | PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: RPS6KA3 | 999 | ALA1201862 | assay format | PubChem BioAssays | ||
9. | ALA1963703 | Functional | PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: PRKCD | 741 | ALA1201862 | assay format | PubChem BioAssays | ||
10. | ALA1963720 | Functional | PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: CHEK2 | 674 | ALA1201862 | assay format | PubChem BioAssays | ||
11. | ALA1963727 | Functional | PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: STK6 | 938 | ALA1201862 | assay format | PubChem BioAssays | ||
12. | ALA1963756 | Functional | PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: MARK3 | 760 | ALA1201862 | assay format | PubChem BioAssays | ||
13. | ALA1963782 | Functional | PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: CHEK1 | 958 | ALA1201862 | assay format | PubChem BioAssays | ||
14. | ALA1963821 | Functional | PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: PDPK1 | 696 | ALA1201862 | assay format | PubChem BioAssays | ||
15. | ALA1963834 | Functional | PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: MARK2 | 646 | ALA1201862 | assay format | PubChem BioAssays | ||
16. | ALA1963835 | Functional | PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: PRKACA | 1,080 | ALA1201862 | assay format | PubChem BioAssays | ||
17. | ALA2033178 | Binding | Inhibition of human recombinant CDK2/CycE using HHASPRK as substrate by ESI-MS analysis | Homo sapiens | 7 | ALA2029332 | protein complex format | Scientific Literature | |
18. | ALA2033179 | Binding | Inhibition of human recombinant ZAP70 using EEEEYEEEE as substrate by ESI-MS analysis | Homo sapiens | 7 | ALA2029332 | single protein format | Scientific Literature | |
19. | ALA2033180 | Binding | Inhibition of human recombinant PYK2 by ESI-MS analysis | Homo sapiens | 7 | ALA2029332 | single protein format | Scientific Literature | |
20. | ALA3430789 | Binding | Delta TM value showing the stabilisation of AMPKA2 produced by compound binding | Homo sapiens | 156 | ALA1145498 | single protein format | Scientific Literature |