| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA949197 | B | Inhibition of VEGFR2 | 24 | single protein format | Scientific Literature | |||
| 2. | ALA949198 | A | Inhibition of human CYP3A4 | Homo sapiens | 17 | single protein format | Scientific Literature | ||
| 3. | ALA949199 | F | Antiproliferative activity against VEGF-stimulated HUVEC | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
| 4. | ALA949200 | A | Inhibition of human CYP1A2 | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 5. | ALA949201 | A | Inhibition of human CYP2C9 | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 6. | ALA949202 | A | Inhibition of human CYP2C19 | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 7. | ALA950138 | A | Inhibition of human CYP2D6 | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 8. | ALA950139 | A | Inhibition of human CYP3A4 using 7-benzyloxy-4-trifluoromethylcoumarin substrate | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 9. | ALA950140 | A | Inhibition of human CYP3A4 using 7-benzyloxyresorufin substrate | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 10. | ALA950141 | A | Metabolic stability in human liver microsomes per mg of protein at 3 uM after 10 mins | Homo sapiens | 3 | microsome format | Scientific Literature | ||
| 11. | ALA950142 | A | Metabolic stability in mouse liver microsomes per mg of protein at 3 uM after 10 mins | Mus musculus | 3 | microsome format | Scientific Literature | ||
| 12. | ALA950143 | A | Cmax in mouse at 50 mg/kg, po | Mus musculus | 3 | organism-based format | Scientific Literature | ||
| 13. | ALA950144 | A | Tmax in mouse at 50 mg/kg, po | Mus musculus | 3 | organism-based format | Scientific Literature | ||
| 14. | ALA950145 | A | AUC (0 to 4 hrs) in mouse at 50 mg/kg, po | Mus musculus | 3 | organism-based format | Scientific Literature | ||
| 15. | ALA950146 | F | Antitumor activity against human L2987 cells xenografted athymic mouse at 30 mg/kg, po administered once daily for 14 days | Homo sapiens | 1 | organism-based format | Scientific Literature | ||
| 16. | ALA950147 | F | Antitumor activity against human L2987 cells xenografted athymic mouse at 90 mg/kg, po administered once daily for 14 days | Homo sapiens | 1 | organism-based format | Scientific Literature | ||
| 17. | ALA950148 | T | Toxicity against human L2987 cells xenografted athymic mouse assessed as occurrence of adverse events at 30 mg/kg, po administered once daily for 14 days | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 18. | ALA950149 | T | Toxicity against human L2987 cells xenografted athymic mouse assessed as occurrence of adverse events at 90 mg/kg, po administered once daily for 14 days | Mus musculus | 1 | organism-based format | Scientific Literature |
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