# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1015630 | B | Inhibition of cow milk xanthine oxidase at 50 ug/mL | Bos taurus | 85 | ALA1150752 | single protein format | Scientific Literature | |
2. | ALA1015631 | B | Inhibition of cow milk xanthine oxidase | Bos taurus | 15 | ALA1150752 | single protein format | Scientific Literature | |
3. | ALA3774271 | B | Inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins followed by substrate addition by FRET assay | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
4. | ALA3774272 | B | Inhibition of human tissue kallikrein-2 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins followed by substrate addition by FRET assay | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
5. | ALA3774273 | B | Inhibition of human tissue kallikrein-3 expressed in baculovirus infected insect cells using Abz-KLYSSQ-EDDnp as substrate preincubated for 10 mins followed by substrate addition by FRET assay | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
6. | ALA3774274 | B | Inhibition of human tissue kallikrein-5 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins followed by substrate addition by FRET assay | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
7. | ALA3774275 | B | Inhibition of human tissue kallikrein-6 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins followed by substrate addition by FRET assay | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
8. | ALA3774276 | B | Inhibition of human tissue kallikrein-7 expressed in baculovirus infected insect cells using Abz-KLYSSQ-EDDnp as substrate preincubated for 10 mins followed by substrate addition by FRET assay | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
9. | ALA3774277 | B | Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate assessed as enzyme Vmax at 2 uM by Lineweaver-Burk plot analysis (Rvb = 450 +/- 20 uM/sec) | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
10. | ALA3774278 | B | Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate assessed as enzyme Vmax at 4 uM by Lineweaver-Burk plot analysis (Rvb = 450 +/- 20 uM/sec) | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
11. | ALA3774279 | B | Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate assessed as enzyme Vmax at 8 uM by Lineweaver-Burk plot analysis (Rvb = 450 +/- 20 uM/sec) | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
12. | ALA3774280 | B | Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate assessed as enzyme Vmax at 10 uM by Lineweaver-Burk plot analysis (Rvb = 450 +/- 20 uM/sec) | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
13. | ALA3774281 | B | Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate assessed as substrate Km at 2 uM by Lineweaver-Burk plot analysis (Rvb = 0.65 +/- 0.03 uM) | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
14. | ALA3774282 | B | Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate assessed as substrate Km at 4 uM by Lineweaver-Burk plot analysis (Rvb = 0.65 +/- 0.03 uM) | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
15. | ALA3774283 | B | Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate assessed as substrate Km at 8 uM by Lineweaver-Burk plot analysis (Rvb = 0.65 +/- 0.03 uM) | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
16. | ALA3774284 | B | Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate assessed as substrate Km at 10 uM by Lineweaver-Burk plot analysis (Rvb = 0.65 +/- 0.03 uM) | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
17. | ALA3774285 | B | Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins followed by substrate addition by Lineweaver-Burk plot analysis | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
18. | ALA3774286 | B | Mixed-type inhibition of human tissue kallikrein-2 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate assessed as enzyme Vmax at 2 uM by Lineweaver-Burk plot analysis (Rvb = 226 +/- 10 uM/sec) | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
19. | ALA3774287 | B | Mixed-type inhibition of human tissue kallikrein-2 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate assessed as enzyme Vmax at 4 uM by Lineweaver-Burk plot analysis (Rvb = 226 +/- 10 uM/sec) | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature | |
20. | ALA3774288 | B | Mixed-type inhibition of human tissue kallikrein-2 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate assessed as enzyme Vmax at 8 uM by Lineweaver-Burk plot analysis (Rvb = 226 +/- 10 uM/sec) | Homo sapiens | 1 | ALA3769311 | cell-based format | Scientific Literature |