# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA644914 | B | The compound was tested in vitro for the inhibition of acetylcholinesterase (AChE) isolated from electric eel at 10e-5 M; NA means no significant activity at 10e-3 M | Electrophorus electricus | 1 | ALA1127171 | single protein format | Scientific Literature | |
2. | ALA644916 | B | The compound was tested in vitro for the inhibition of acetylcholinesterase (AChE) isolated from electric eel at 10e-6 M; NA means no significant activity at 10e-3 M | Electrophorus electricus | 1 | ALA1127171 | single protein format | Scientific Literature | |
3. | ALA650964 | B | Displacement of [3H]flunitrazepam from GABA-A benzodiazepine receptor (BZR) of rat brain membranes (NA = no significant activity) | Rattus norvegicus | 1 | ALA1127171 | cell membrane format | Scientific Literature | |
4. | ALA651676 | B | Binding affinity for rat GABA-A Benzodiazepine receptor inverse agonist site | Rattus norvegicus | 1 | ALA1129323 | protein complex format | Scientific Literature | |
5. | ALA649962 | B | In vitro inhibition of [3H]flunitrazepam binding to GABA-A receptor of rat cerebral cortex membranes | 9 | ALA1124604 | cell membrane format | Scientific Literature | ||
6. | ALA858255 | B | Binding affinity towards benzodiazepine receptor inverse agonist site by the displacement of [3H]diazepam in rat cerebral cortical membranes. | 51 | ALA1126835 | cell membrane format | Scientific Literature | ||
7. | ALA650289 | B | In vitro inhibition of 3[H]Diazepam binding to Benzodiazepine receptor from rat cerebral cortical membranes | 43 | ALA1125077 | cell membrane format | Scientific Literature | ||
8. | ALA652555 | B | Hill coefficient for inhibition of ~2 nM [3H]diazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortical membrane | 5 | ALA1122149 | assay format | Scientific Literature | ||
9. | ALA652562 | B | In vitro inhibition of [3H]diazepam binding to benzodiazepine receptor in rat cerebral cortical membrane | 48 | ALA1122149 | cell membrane format | Scientific Literature | ||
10. | ALA650178 | B | In vitro inhibition of binding to the benzodiazepine receptor in rat cerebral cortical membrane using [3H]diazepam as radioligand | Rattus norvegicus | 18 | ALA1124212 | cell membrane format | Scientific Literature | |
11. | ALA650464 | B | Displacement of [3H]-diazepam from GABA-A benzodiazepine receptor of rat cerebral cortex | Rattus norvegicus | 6 | ALA1123687 | tissue-based format | Scientific Literature | |
12. | ALA653130 | B | In vitro inhibition of [3H]diazepam binding to rat cerebral cortical membrane benzodiazepine receptors | 22 | ALA1122642 | assay format | Scientific Literature | ||
13. | ALA650075 | B | Inhibition on Benzodiazepine receptor | 43 | ALA1130277 | protein complex format | Scientific Literature | ||
14. | ALA652650 | B | Affinity to displace [3H]flunitrazepam from Benzodiazepine receptor in bovine brain membrane | 21 | ALA1125055 | cell membrane format | Scientific Literature | ||
15. | ALA651487 | B | Concentration that inhibits specific [3H]flunitrazepam binding to benzodiazepine receptor in bovine brain | 19 | ALA1122458 | assay format | Scientific Literature | ||
16. | ALA652195 | B | In vivo inhibition of specific [3H]flunitrazepam binding in mouse brain 10 minute after iv administration of 15 uM/Kg | Mus musculus | 12 | ALA1122458 | organism-based format | Scientific Literature | |
17. | ALA653049 | B | In vitro displacement of [3H]flunitrazepam from GABA-A central benzodiazepine receptor of rat cerebral cortex membranes | Rattus norvegicus | 8 | ALA1128336 | cell membrane format | Scientific Literature | |
18. | ALA653051 | B | In vitro binding affinity at benzodiazepine receptor of rat cerebral cortical membranes by [3H]diazepam displacement. | Rattus norvegicus | 18 | ALA1125333 | assay format | Scientific Literature | |
19. | ALA657475 | B | Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brain | Cavia porcellus | 18 | ALA1126472 | assay format | Scientific Literature | |
20. | ALA663495 | B | Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreas | 18 | ALA1126472 | assay format | Scientific Literature |