| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA963295 | F | Agonist activity at NTR1 expressed in CHOK1 cells assessed as stimulation of calcium mobilization at 10 uM relative to neurotensin | 14 | cell-based format | Scientific Literature | |||
| 2. | ALA963296 | F | Agonist activity at NTR1 expressed in CHOK1 cells by calcium mobilization assay | 8 | cell-based format | Scientific Literature | |||
| 3. | ALA963297 | F | Agonist activity at NTR1 expressed in CHOK1 cells by calcium mobilization assay relative to neurotensin | 8 | cell-based format | Scientific Literature | |||
| 4. | ALA3101314 | F | Ratio of EC50 for NTR1 in human U2OS cells to EC50 for NTR1 (unknown origin) expressed in CHO cells assessed as Ca2+ mobilization | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 5. | ALA3101317 | B | Inhibition of MOR (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA3101318 | B | Inhibition of DOR (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA3101828 | A | Cytotoxicity in human Fa2N-4 cells after 24 hrs | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 8. | ALA3101829 | A | Metabolic stability in mouse liver microsomes assessed as compound remaining at 1hr | Mus musculus | 3 | microsome format | Scientific Literature | ||
| 9. | ALA3101830 | A | Metabolic stability in human liver microsomes assessed as compound remaining at 1 hr | Homo sapiens | 3 | assay format | Scientific Literature | ||
| 10. | ALA3101831 | A | Metabolic stability in human plasma assessed as compound remaining at 3 hrs | Homo sapiens | 3 | cell-free format | Scientific Literature | ||
| 11. | ALA3101832 | A | Metabolic stability in mouse plasma assessed as compound remaining at 3 hrs | Mus musculus | 3 | cell-free format | Scientific Literature | ||
| 12. | ALA3101833 | A | Plasma protein binding in mouse at 10 uM | Mus musculus | 3 | cell-free format | Scientific Literature | ||
| 13. | ALA3101834 | A | Plasma protein binding in human at 10 uM | Homo sapiens | 3 | cell-free format | Scientific Literature | ||
| 14. | ALA3101937 | A | Plasma protein binding in mouse at 1 uM | Mus musculus | 3 | cell-free format | Scientific Literature | ||
| 15. | ALA3101938 | A | Blood brain permeability of the compound at donor and acceptor pH 7.4 by PAMPA | 3 | tissue-based format | Scientific Literature | |||
| 16. | ALA3101939 | A | Plasma protein binding in human at 1 uM | Homo sapiens | 3 | cell-free format | Scientific Literature | ||
| 17. | ALA3101940 | B | Inhibition of DAT (unknown origin) | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 18. | ALA3101941 | B | Inhibition of NTS1 receptor (unknown origin) | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 19. | ALA3101942 | A | Permeability of the compound at donor and acceptor pH 7.4 by PAMPA | 3 | assay format | Scientific Literature | |||
| 20. | ALA3101943 | A | Permeability of the compound at donor pH 6.2 and acceptor pH 7.4 by PAMPA | 3 | assay format | Scientific Literature |
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