| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA715566 | B | Negative logarithm of relative affinity (pRA) towards melatonin receptor (relative to N-acetyl-5-methoxytryptamine (aMT)) | Coturnix | 132 | ALA1131632 | protein format | Scientific Literature | |
| 2. | ALA874168 | B | inhibitory concentration against Melatonin receptor | Coturnix | 17 | ALA1131632 | protein format | Scientific Literature | |
| 3. | ALA714927 | B | Binding affinity for Melatonin receptor using 2-[125I]iodomelatonin as radioligand | Coturnix | 17 | ALA1131632 | protein format | Scientific Literature | |
| 4. | ALA714100 | F | Intrinsic activity evaluated on [35S]GTP-gamma-S, binding in NIH3T3 cells stably transfected with human Melatonin receptor type 1A | 3 | ALA1136758 | cell-based format | Scientific Literature | ||
| 5. | ALA715950 | B | Relative Binding Affinity (pRA1) to cloned human Melatonin receptor type 1A, stably expressed in NIH3T3 rat fibroblast cells, determined using 2-[125I]iodomelatonin | 4 | ALA1136758 | cell-based format | Scientific Literature | ||
| 6. | ALA715953 | B | Binding Affinity (pKi) towards Melatonin receptor type 1A | 1 | ALA1136758 | single protein format | Scientific Literature | ||
| 7. | ALA710593 | F | Intrinsic activity evaluated on [35S]GTP-gamma-S, binding in NIH3T3 cells stably transfected with human Melatonin receptor type 1B | 3 | ALA1136758 | cell-based format | Scientific Literature | ||
| 8. | ALA713142 | B | Relative Binding Affinity (pRA1) to cloned human Melatonin receptor type 1B, stably expressed in NIH3T3 rat fibroblast cells, determined using 2-[125I]iodomelatonin | 4 | ALA1136758 | cell-based format | Scientific Literature | ||
| 9. | ALA858415 | B | Binding Affinity (pKi) towards human Melatonin receptor type 1B | 4 | ALA1136758 | single protein format | Scientific Literature | ||
| 10. | ALA839211 | B | Ratio of IC50 to that IC50 aMT (aMT=melatonin N-acetyl-5-methoxytryptamine) | Coturnix | 17 | ALA1131632 | single protein format | Scientific Literature | |
| 11. | ALA839735 | B | Inhibition of 2-[125I]iodomelatonin binding to human melatonin receptor MT2 expressed in NIH3T3 rat fibroblast cells | Homo sapiens | 10 | ALA1139541 | cell-based format | Scientific Literature | |
| 12. | ALA838521 | B | Inhibition of 2-[125I]iodomelatonin binding to human melatonin receptor type 1A (MT1) expressed in NIH3T3 rat fibroblast cells | Homo sapiens | 11 | ALA1139541 | cell-based format | Scientific Literature |
The page will load shortly, Thanks for your patience!